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N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3-methoxypiperidine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-methoxy-N-(pyridin-3-ylmethyl)propanamide
3,4,7-trimethyl-2-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-1H-indole
1-{3-oxo-3-[3-(2-phenylacetyl)piperidin-1-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[1-(2-chlorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}methanesulfonamide
2-{4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperazin-1-yl}acetic acid
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
(2R,3R,6R)-5-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[2-(piperidin-1-yl)ethyl]propanamide
1-tert-butyl-4-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)piperidin-2-one
3,5-dimethyl-1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}-1H-pyrazole
5-[3-(3-phenylpropanoyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-[2-(4-methylmorpholin-2-yl)ethyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
4-benzyl-3-[1-(2-oxo-1,3-oxazolidine-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[4-(4-{[2-(1H-indol-3-yl)ethyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
4-(3-{[3-(3-methylphenyl)phenyl]carbamoyl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
1-(2-methyl-1H-1,3-benzodiazol-6-yl)-3-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}urea
methyl 2-(cyclohexylsulfamoyl)-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-butyl-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
8-(3-chloro-4-hydroxybenzoyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{2-chloro-4-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]phenoxy}acetamide
1-methyl-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
1-(2,3-difluoro-6-methoxybenzoyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
(3R,4S)-4-phenyl-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidin-3-amine
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
(3S,4S)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
2-(furan-2-yl)-N-[4-(1H-pyrazol-1-yl)phenyl]azepane-1-carboxamide
3-amino-2-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazine-1-carboxamide
3,5,7-trimethyl-N-[3-(4-methylpiperazin-1-yl)butyl]-1H-indole-2-carboxamide
2-methyl-2-(2-{7-methyl-2,7-diazaspiro[4.4]nonan-2-yl}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-[benzyl({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]propanamide
2-(azocan-1-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(3-methoxybenzoyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
N3-[(2-chloropyridin-3-yl)methyl]-N3-methylpiperidine-1,3-dicarboxamide
5-propyl-4-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine
methyl 1-{[(1-ethyl-1H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-pyrazole-3-carboxylate
2-(4-methylphenyl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyrimidin-4-ol
5-(2-methoxyphenoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{5-[3-(1H-pyrazol-3-yl)phenyl]furan-2-carbonyl}morpholine
8-(2H-1,3-benzodioxole-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
3,3,3-trifluoro-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]propanoic acid
3-(3,4-dimethoxybenzoyl)-1-(propane-2-sulfonyl)piperidine