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1-(3,4-dimethylphenyl)-N-[(5-methylthiophen-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[2-(2-phenylethyl)morpholin-4-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-(3-methyl-1H-pyrazol-1-yl)-N-[(3-methyl-1H-pyrazol-5-yl)methyl]propanamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(2-ethoxyacetyl)pyrrolidine-3-carboxylic acid
2-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)pyridine
1-(2-chloropyridin-3-yl)-3-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
2-(2,4-dichlorophenoxy)-N-(2-methanesulfonylethyl)acetamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-[2-(methylsulfanyl)pyridine-3-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
4-(cyclohex-3-en-1-yl)-1-[2-(pyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-tert-butyl-N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-4-hydroxypyrimidine-5-carboxamide
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidine
1-[2-oxo-2-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)ethyl]pyrrolidin-2-one
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(3-methoxyphenyl)methyl]-N-(3-methoxypropyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-4-{[(4-methylphenyl)amino]methyl}benzamide
1-(4-fluorophenyl)-2-(4,4,4-trifluorobutyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(4aS,8aR)-6-[(2-methyl-1H-imidazol-4-yl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]propanamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-(2-ethoxyacetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-2-{3-oxo-2-azaspiro[4.5]decan-2-yl}-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
6-({3-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
N-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N,3-dimethyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-3,4-dihydrophthalazine-1-carboxamide
(2S,4R)-4-(cyclooctylamino)-1-[(2,3-dimethoxyphenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
2-[2-(9-ethyl-9H-carbazol-3-yl)-1H-imidazol-1-yl]propane-1,3-diol
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(1,3-thiazol-2-yl)piperazine
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
1-(6-aminopyrimidin-4-yl)-4-(1H-imidazol-2-ylmethyl)-1,4-diazepane-6-carboxylic acid
2-(pyridin-2-yl)-5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}pyrimidine
methyl 3-(2-methoxybenzoyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(cyclohexylsulfamoyl)-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(1H-pyrazol-3-yl)benzamide
N,2-dicyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)quinoline-4-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(1H-1,2,4-triazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-tert-butyl-6-[(3,4-dimethylpiperazin-1-yl)methyl]phenol
3-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methoxy}pyridin-2-amine
ethyl 1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-(2-methoxyethyl)piperidine-3-carboxylate
3-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}pyridin-2-amine
2-(1H-imidazol-1-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
1-[(5-methylfuran-2-yl)methyl]-3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
1-(4-{[4-(4-methoxyphenoxymethyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-N'-methyl-N'-[1-(thiophen-2-yl)ethyl]ethanediamide
2-amino-4-[6-(dimethylamino)pyridin-3-yl]-6-hydroxy-5H-indeno[1,2-b]pyridine-3-carbonitrile
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methoxyphenyl)propan-1-one
2-(2,4-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one