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N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-methyl-3-(3-methylpiperidin-1-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-methyl-6-{5-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
5-(4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-[2-(trifluoromethyl)phenyl]pyrimidine
5-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
3-methyl-1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}butan-1-one
2-{[4-(adamantan-2-yl)piperazin-1-yl]methyl}-4-(6-methoxypyridin-2-yl)phenol
N-methyl-3-phenyl-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
2-(1-benzyl-1H-pyrazol-4-yl)-4-(pyrrolidine-1-carbonyl)pyridine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[2-(oxan-2-yl)ethyl]propanamide
2-[6-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-methylpyrimidin-4-yl]ethan-1-amine
N-{1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(3-{2-[1-(3-fluoropyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-{1-[4-(4-fluorophenoxy)piperidin-1-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
1-[6-chloro-3-(1,4-oxazepan-4-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]azocane
4-[1-(3-methylbutyl)-5-[4-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-[4-(2,3-dimethylphenyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
6-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-2,4-dimethylpyridine-3-carbonitrile
3-{5-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-ethyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-4-carboxamide
8-methoxy-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-{[4-(morpholin-4-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
N-(1-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
(3R,4S)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3,4-dimethylpiperidin-4-ol
4-phenyl-5-propyl-1-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-imidazole
3-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}-6-methyl-4H-chromen-4-one
2-benzyl-N-(2,3-dihydro-1H-inden-2-yl)-1,3-benzoxazole-5-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-3,5-dimethyl-1H-indole-2-carboxamide
4-[(5-butylthiophen-2-yl)methyl]-2-(trifluoromethyl)morpholine
6-chloro-2-{2-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
1-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
1-{2-[2-(4-methanesulfonylphenyl)phenoxy]ethyl}-1H-imidazole
2-(2-propyl-1,3-thiazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3S,7S)-5-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-methylpiperidine
2-(4-methanesulfonylphenyl)-1-(2-phenoxyethyl)-1H-imidazole
5-methyl-3-{[methyl({2-[(4-methylphenyl)sulfanyl]ethyl})amino]methyl}-1H-indole-2-carboxylic acid
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[3-(pyridin-3-yl)propyl]-1H-pyrazole-4-carboxamide
3-(3-fluorophenyl)-4-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-pyrazole
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-(pyridin-2-yl)prop-2-enamide
(2S)-2-amino-1-[7-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]pentan-1-one
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}furan-2-carboxamide
3-benzyl-4-(2,4,5-trifluorobenzoyl)piperazin-2-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}piperidine-4-carboxamide
1-(2-{[(8-chloroquinolin-5-yl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
1-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-4-(4-fluorophenyl)butane-1,4-dione