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2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-cycloheptyl-N-methyl-2-phenylacetamide
8-(2-methyl-5-propylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
6-[2-(4-methylphenoxy)acetyl]-N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[1-(2,2,2-trifluoroethyl)-1H-imidazol-2-yl]pyridine
1-{4-[4-(4-methoxyphenoxy)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-[1-(2,3-dihydro-1H-inden-4-yl)-5-{5-[(dimethylamino)methyl]furan-2-yl}-1H-1,2,4-triazol-3-yl]acetamide
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(2,2-dimethyloxan-4-yl)-1H-pyrazole-4-carboxamide
3-(4-fluoro-2-methylphenyl)-1-[(3R)-piperidin-3-yl]urea
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl][(4-phenyl-1,3-thiazol-2-yl)methyl]amine
1-{1'-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-(4-methylphenyl)-2-({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)propanamide
4-(2-chloro-6-methoxyphenyl)-2-ethyl-6-methylpyrimidine
4-{4-[4-(2-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[4-(4-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-(4-methoxyphenyl)acetamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(4-methoxypyrimidin-2-yl)piperazin-2-yl}ethan-1-ol
4-{1,1-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-(3-methoxyphenoxymethyl)-1,3-oxazole
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
5-(2-{[(3-methylphenyl)methyl]amino}ethyl)-1-(prop-2-en-1-yl)pyrrolidin-2-one
methyl 4-{[(4aR,8aS)-1-(2-methoxy-2-phenylacetyl)-decahydro-1,6-naphthyridin-6-yl]methyl}benzoate
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-5,7-dimethyl-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
(3S,7S)-5-[2-(azepan-1-yl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-amino-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,6-dimethyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[4-(2-hydroxyethyl)phenyl]-5-[1-(oxan-4-yl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
6-methyl-5-(5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
5-(3,5-difluoro-4-methoxyphenyl)-1-[(2S)-1-methoxypropan-2-yl]-4-phenyl-1H-imidazole
1-[(4-hydroxy-3,5-dimethylphenyl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
3-[(2R,3R,6R)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(3S,4R)-1-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
5-(2-chlorophenyl)-N-[(3R,4R)-4-hydroxypiperidin-3-yl]furan-2-carboxamide
2-amino-4-(3,4-dihydroxyphenyl)-7-methoxy-5H,6H-benzo[h]quinoline-3-carbonitrile
4-[(4-chlorophenyl)methyl]-1-methylpiperazine-2-carboxylic acid
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-(methoxymethyl)-N-{[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}furan-2-carboxamide
1-methyl-9-(3-methyl-1H-pyrazole-5-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
2-cyclopropyl-3-oxo-N-(2-phenylethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(3,5-difluoro-2-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-1-{1-oxaspiro[4.4]nonan-3-yl}-1H-imidazole
ethyl 5-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-{[4-(2-methylphenoxy)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
2,4-dimethyl-N-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)benzamide
methyl 1-(2-methoxyethyl)-3-(3-methylbutanamido)-5-[(5-methylhex-5-en-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(1-cyclohexylpiperidine-4-carbonyl)-3-(1H-imidazol-4-ylmethyl)piperazin-2-one
6-methyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}pyridazin-3-amine
3-(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)propanamide
2-(furan-2-yl)-5-(1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-imidazol-2-yl)pyrimidine
1-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
N-[2-({1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)ethyl]acetamide