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N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methyl-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanamide
5-ethyl-N-[(2-methoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(4S)-3,3,4-trimethyl-1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-ol
(4aS,8aR)-6-(furan-3-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidin-3-yl)piperazine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
N-ethyl-1-[2-(piperazin-1-yl)ethyl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}quinoxaline-5-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
5-propyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
methyl 4-methoxy-3-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)benzoate
3-methyl-7-{[3-(pyridin-2-yl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-({[(3R,4R)-1-[(3-chloro-1-benzothiophen-2-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-(1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-1,2,3-triazol-4-yl)phenol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
[(3S,5R)-1-(1-benzothiophen-2-ylmethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
9-(cyclopropylmethyl)-1-methyl-4-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(5-acetamido-1H-1,2,4-triazol-3-yl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
7-methanesulfonyl-N,4-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}quinazolin-2-amine
6-[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyrazine-2-carboxamide
5-[1-(2-ethylbutyl)-4-hydroxypiperidin-4-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
6-hydroxy-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-1,4-oxazepane-4-carboxamide
(3R,4R)-1-(2-amino-6-methoxypyrimidin-4-yl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
N-[2-(furan-2-yl)ethyl]-4-sulfamoylbenzamide
N-cyclopropyl-N-({5,8-dimethoxy-2-[methyl(thiophen-2-ylmethyl)amino]quinolin-3-yl}methyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-(5-{[cyclopropyl(pyridin-3-ylmethyl)amino]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-ethyl-5-methoxy-1-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-indole-2-carboxamide
1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-4-benzyl-3-ethyl-1,4-diazepan-5-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-methyl-3-[(oxolan-3-yl)sulfamoyl]-N-(thian-4-yl)benzamide
N-tert-butyl-2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
4-ethyl-3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-1-(3,5-dimethoxybenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
2-{5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
(3R,4R)-4-amino-1-{[3-(4-fluorophenoxy)phenyl]methyl}piperidin-3-ol
4-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,5-dimethyl-1H-pyrazole
3-[3-(methylsulfanyl)phenyl]-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
3-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine
(2S,4R)-N-ethyl-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamido]-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
N-(4-methoxy-2-methylphenyl)-3-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}propanamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-ethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-(3-{[(1-methanesulfonylpiperidin-4-yl)amino]methyl}-1H-indol-1-yl)propanamide
5-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
2-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}-6-methoxyphenol
3-(2-amino-1,3-thiazol-4-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
N-[5-chloro-2-(2-methylpiperidin-1-yl)phenyl]-3-(1,2-oxazolidin-2-yl)propanamide
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(propan-2-yloxy)benzamide
3-(3-fluorophenyl)-4-[3-(1,2-oxazolidin-2-yl)propanoyl]piperazin-2-one