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5-[2-(3-fluorophenyl)piperidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-(1,4-diazepane-1-carbonyl)-6-(4-methoxyphenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-(3-methoxyphenyl)-5-(2-methyloxolane-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(2-chloro-4-fluorophenyl)-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-5-phenyl-1,2-oxazole-4-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(2-fluorophenyl)methyl](oxolan-2-ylmethyl)amine
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-3-propanamidobenzamide
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
6-(2,3-dichlorophenyl)-N,N-dimethylpyridazin-3-amine
2-{[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]methyl}benzoic acid
2-ethyl-1-methyl-4-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
1-[(3,5-dimethoxyphenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
(3S,5S)-1-(3-methylbut-2-en-1-yl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
2-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}-6-methylpyridin-3-ol
ethyl 4-(3-{2-[(3-chloro-4-methoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)piperidine-1-carboxylate
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(3-methoxyphenoxymethyl)piperidine
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
[3-(cyclopropylmethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl]methanol
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1,3-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(4-methoxypiperidin-1-yl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
4-[1-(3-methylbutyl)-5-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
(3R,4S)-4-cyclopropyl-1-(3-fluoro-4-methylbenzenesulfonyl)pyrrolidin-3-amine
[4-(5-methyl-4-phenylthiophene-3-carbonyl)-1,4-oxazepan-6-yl]methanol
3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
N-[3,3-dimethyl-1-(pyrrolidin-1-yl)butan-2-yl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
4-[(2-methoxyethyl)amino]-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
8-(dimethyl-1,3-oxazole-5-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
methyl 3-[(3S,4R)-1-[(4-methoxynaphthalen-1-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoate
ethyl 1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decane-8-carboxylate
3-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
6-methoxy-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrimidin-4-amine
5-cyclopropanecarbonyl-1'-(dimethyl-1,3-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(4-fluorophenyl)methyl]-1-[(1-methyl-1H-pyrazol-5-yl)methyl]piperidine
N-(4-fluorophenyl)-4'-(2-methoxyethyl)-3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-carboxamide
N-(2-phenylethyl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine-4-carboxamide
3-ethyl-1-[2-(pyrrolidin-1-yl)benzoyl]piperidine-3-carboxylic acid
2-[4-(1-cyano-1-methylethyl)phenyl]-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
N-(isoquinolin-5-ylmethyl)-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
1-{6-[5-chloro-2-(propan-2-yloxy)phenyl]pyridin-2-yl}ethan-1-ol
2-(3-methyl-1,2-oxazol-5-yl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
3-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{methyl[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}propanamide
(2E)-3-(3,4-dimethoxyphenyl)-N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)prop-2-enamide
2-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyridine-3-carboxylic acid
2-amino-4-(1H-indol-3-yl)-6-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
[1-({[1-(3-methoxyphenyl)propan-2-yl]amino}methyl)cyclopentyl]methanol
8-chloro-2-({3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)quinoline
N-ethyl-2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}acetamide