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{6-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyridin-2-yl}methanol
3-(4-methoxyphenyl)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
4-(4-{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-6-ethylpyrimidine
2-{4-[(5-phenylthiophen-2-yl)methyl]morpholin-3-yl}acetic acid
1-ethyl-4-[3-(1H-imidazol-2-yl)benzoyl]-2,2-dimethylpiperazine
6-{4-hydroxy-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine-1-carbonyl}piperazin-2-one
N-cyclopentyl-3-{5-[2-(methylsulfanyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrazine
N-cyclopropyl-N-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
4-[2-(dimethylamino)-6-(trifluoromethyl)pyrimidin-4-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl][1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
1-(2,6-diaminopyrimidin-4-yl)-3-(3-phenylpropyl)piperidine-3-carboxylic acid
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2-methoxyethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
6-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}-1H-indazole
2-cyclopropyl-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-[4-(2-methoxyethoxy)phenyl]-5-(pyrrolidin-1-ylmethyl)pyridine
(1s,4s)-4-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]cyclohexan-1-ol
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-N-(2-phenylethyl)acetamide
(2R)-1-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)pyrrolidine-2-carboxamide
(1r,4r)-4-[(4-ethoxypyrimidin-2-yl)amino]cyclohexan-1-ol
N-[(3S,4R)-1-(dimethylsulfamoyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-3-methoxypyrazine
2-chloro-4-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]benzamide
(3-{2-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(morpholin-4-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]cyclohexane-1-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(pyridin-2-ylmethyl)acetamide
2-{2-[1-(2,5-dichlorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
1-({5-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-cyclopentyl-1-(3-methylbutyl)-4-oxo-5-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
5-fluoro-2-[(2-methoxyphenyl)methyl]-1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
1-(2-chlorophenyl)-3-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methylurea
1-[2-(1-tert-butyl-3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]piperidine-4-carboxamide
9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3,3-bis(hydroxymethyl)-N-[2-(3-methylphenoxy)phenyl]piperidine-1-carboxamide
N,1,6-trimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[4-(dimethyl-1,2-oxazol-4-yl)phenyl]pyrimidin-5-ol
(3S,4S)-1-{[4-(furan-2-yl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
3-(4-methylphenyl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
1-tert-butyl-3-cyclopropyl-5-[(2-methylphenyl)methyl]-1H-1,2,4-triazole
N-(2-{4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]phenoxy}ethyl)acetamide
2-[2-methyl-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]pyridine
2-{2-[(4-methoxypiperidin-1-yl)methyl]-4-(pyridin-3-yl)phenoxy}acetic acid
5-{5-acetyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
(3aS,6aS)-2-cyclopentanecarbonyl-5-(1H-indol-7-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine