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(3aS,6aR)-3-[2-(pyridin-2-yl)ethyl]-5-(thian-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
7-(5-chloro-2-methoxyphenyl)-4-[(4-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,3,5-trimethyl-N-(pyrazin-2-ylmethyl)-1-benzofuran-2-carboxamide
N,4-dimethyl-2-(propan-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-5-carboxamide
2-{4-[4-(thiomorpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
1-{5-[(4-hydroxyphenyl)methyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,4-diazepan-5-one
3-(4-methyl-1H-pyrazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
N-cyclohexyl-N-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
4-(3,5-difluoropyridine-2-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
[(3-chloropyridin-4-yl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
3-(1-ethyl-1H-pyrazol-5-yl)-1-{3-[(pyridin-3-yl)amino]propyl}urea
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetic acid
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3,4-dimethylphenoxy)ethan-1-one
4-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
2-[3-(1H-indol-3-yl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
4-(1H-imidazol-1-ylmethyl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-ol
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(propan-2-yl)piperidine-3-carboxamide
2-ethyl-4-methyl-N-(2-propoxypropyl)-1,3-oxazole-5-carboxamide
N-(3-cyano-4-methylphenyl)-3-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide
N-(furan-3-ylmethyl)-N-methyl-2-(1H-pyrazol-1-yl)butanamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-2-(pyridin-3-yl)acetamide
2-[5-(methoxymethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]-6-methylpyridine
(2S,5R)-2,5-dimethyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-4-(2-oxopiperidin-1-yl)butanamide
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(pyridin-2-ylmethyl)acetamide
N-(3-methoxyphenyl)-3-[2-(2,2,3,3-tetrafluoropropoxy)acetamido]benzamide
[3-(cyclopropylmethyl)-1-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidin-3-yl]methanol
N-{3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-4-methylbenzamide
7-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-amino-4-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-(3-benzylphenyl)-3-oxo-2-(propan-2-yl)piperazine-1-carboxamide
N-{[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
4-{4-phenyl-1-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-imidazol-5-yl}pyridine
N-[4-(3-methoxyphenyl)phenyl]-1-(2-oxopropanoyl)piperidine-3-carboxamide
2-[2-(2-amino-3-cyano-6-cyclopropylpyridin-4-yl)-4-chlorophenoxy]acetic acid
2-{[(3R,4S)-3-amino-4-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}-6-fluoroquinolin-4-ol
2-ethyl-4-methyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1,3-oxazole-5-carboxamide
(1R,5S,6R)-6-{[4-(4-methylbenzenesulfonyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
2-[4-(cyclopropylmethoxy)phenyl]-2-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]acetic acid
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]piperidin-2-one
2-(1-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-imidazol-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
N-(butan-2-yl)-2-(difluoromethoxy)-N-(pyridin-4-ylmethyl)benzamide
2-(5-chloropyridine-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one