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5-[1-(1-benzylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]-N-(propan-2-yl)pyrimidin-2-amine
4-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
2-[(prop-2-en-1-yl)amino]-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-chloro-4-[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]benzamide
4-(dimethyl-1,3-thiazole-5-carbonyl)-N-(2-fluorophenyl)morpholine-2-carboxamide
1-[2-({[4-(pyridin-3-yl)pyrimidin-2-yl]amino}methyl)morpholin-4-yl]ethan-1-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[2-(dimethylamino)-4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-3,3-dimethylbutan-1-one
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylbutan-1-one
(furan-3-ylmethyl)({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
1-[(2-carboxyphenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
(4aS,8aR)-6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
3-chloro-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-5-(trifluoromethyl)pyridin-2-amine
1-{4-[4-(2-amino-1,3-benzothiazole-5-carbonyl)piperazin-1-yl]phenyl}ethan-1-one
4-benzyl-3-ethyl-1-[2-(methylamino)benzoyl]-1,4-diazepan-5-one
4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
1-({4-[(5-acetamidothiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-N,N-diethylpiperidine-3-carboxamide
3-amino-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole-5-carboxamide
5-[(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)methyl]-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(5-methylfuran-2-yl)-N-[2-(2-methylpropanesulfonyl)ethyl]benzamide
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]propanamide
2-cyclopropyl-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]pyrimidine-5-carboxamide
propan-2-yl 2-[(7-fluoro-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
2-methyl-5-[4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
methyl 3-(cyclobutylmethoxy)-5-{[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}benzoate
(3S,4R)-N,N-dimethyl-4-propyl-1-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]pyrrolidin-3-amine
N,N-dimethyl-7-(2-methyloxolane-2-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2R)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}oxolane-2-carboxamide
2-(5-acetylthiophen-3-yl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}acetamide
N-(1-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
N-[(3R,4S)-1-(2-ethoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(pyridin-3-yl)acetamide
1-(3,5-dimethylphenyl)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
1-benzyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,4-diazepan-6-ol
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
1-{2-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-phenylpropan-1-one
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-[2-methyl-2-(morpholin-4-yl)propyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-(cyclobutylmethyl)-3-({[(3-fluoro-4-methylphenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
[(2-ethylpyrimidin-4-yl)methyl](methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
2-(4-methanesulfonylphenyl)-6-methylpyridine-3-carbonitrile
2-methoxy-1-{4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
N-{4-[2-(1H-imidazol-4-yl)acetamido]phenyl}pentanamide
4-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)butanamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
7-methanesulfonyl-4-methyl-2-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-1-yl]quinazoline
2-({[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)ethan-1-ol
(1R,3S)-3-amino-N-[(3-chlorophenyl)methyl]-N-cyclopropylcyclohexane-1-carboxamide
9-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(4-methoxyphenyl)-4-oxobutanamide
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine