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1-[2-(4-chlorophenyl)morpholine-4-carbonyl]cyclopropan-1-amine
N-[3-(furan-2-yl)phenyl]-1-(4-oxo-4H-chromene-2-carbonyl)piperidine-4-carboxamide
N-methyl-1-(pyridine-2-carbonyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)piperidine-4-carboxamide
ethyl 4-[2-(3,4-dichlorophenyl)morpholin-4-yl]butanoate
1-(cyclohexylmethyl)-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
2,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-(2-fluoro-4-methylphenyl)-3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
[1-(6-cyclopropylpyrimidin-4-yl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-ethyl-4-{[4-methyl-4-(methylsulfanyl)pentan-2-yl]amino}piperidine-1-carboxamide
3-methyl-8-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
8-{3-cyclopropyl-5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}quinoline
N'-cycloheptyl-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}butanediamide
3-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]propanoic acid
(2S,4S)-N-ethyl-4-(furan-2-amido)-1-(2-methanesulfonylacetyl)pyrrolidine-2-carboxamide
1-cyclopentyl-4-[4-(4-methylpyridin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
2-(2-chlorophenyl)-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
2-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
3,3-dimethyl-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-1H-1,2,4-triazole-5-carboxamide
N-[(3S,4R)-1-(5-oxo-5-phenylpentanoyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-(1H-1,2,3-benzotriazol-4-yl)-1-(1-methanesulfonylpiperidin-4-yl)urea
N-[2-(N-methylmethanesulfonamido)ethyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(2R,6R)-4-[2-(4-hydroxyphenyl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
(3S,4S)-4-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-1-(propan-2-yl)pyrrolidin-3-ol
1,3-dimethyl-6-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[2-({4-[ethyl(methyl)amino]pyrimidin-2-yl}oxy)hex-5-en-1-yl](methyl)amino}-N,N-dimethylacetamide
3-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}piperidin-2-one
4-[(4-methylphenyl)methyl]-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]piperazin-2-one
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-methoxypropyl)piperidine
N-[2-(benzyloxy)ethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
N-{[3-methyl-7-(2-oxo-2-phenylacetyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
N-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)-6-methylpyridine-3-carboxamide
N5-cyclooctyl-N3-(cyclopropylmethyl)-4-oxo-1-(oxolan-2-ylmethyl)-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
3-({[2-(2-fluorophenyl)ethyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]piperidine-4-carboxylic acid
1-methyl-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-indazole
1-(2-aminoethyl)-N-(1-cyclopentanecarbonylazepan-3-yl)-1H-1,2,3-triazole-4-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(4-fluorophenyl)propan-1-one
5-propyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
[2-(dimethylamino)ethyl]({2-[(6-methoxypyrimidin-4-yl)oxy]hex-5-en-1-yl})methylamine
1-[7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-(3-methylbutyl)-8-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(azepan-1-yl)-1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
2-(2,4-difluorophenyl)-2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]acetic acid
3-(2-chlorophenyl)-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]propan-1-one
2,6-dimethoxy-3-[5-(pyridin-4-yl)-1H-pyrazol-4-yl]pyridine
3-(5-{4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid