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2,8-dimethyl-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}quinoline
(2S,4R)-4-amino-N,N-diethyl-1-[2-(pyridin-4-yl)acetyl]pyrrolidine-2-carboxamide
6-methyl-N-[3-(4-methylpiperazin-1-yl)butyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-(3-methoxypropyl)-8-(4-methylpyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-ethyl-4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4,6-dimethyl-2-{methyl[2-(morpholin-4-yl)propyl]amino}pyridine-3-carboxamide
1-(2-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-2,3-dihydro-1H-inden-2-yl)piperidine
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
N-(furan-2-ylmethyl)-2-{4-[3-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-N-methyl-6-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-(propan-2-yl)pyridazine
3-methyl-1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
7-{[ethyl(oxan-4-ylmethyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-[(2S,4R,6S)-2-[2-(methoxymethyl)pyrimidin-5-yl]-6-(2-phenylethyl)oxan-4-yl]acetamide
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
5-({3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}methyl)-2-hydroxybenzoic acid
N-ethyl-2,8-dimethyl-N-(oxolan-2-ylmethyl)quinoline-4-carboxamide
2-(2-fluorophenoxymethyl)-N-methyl-N-(quinolin-4-ylmethyl)-1,3-oxazole-4-carboxamide
1-ethyl-N-[3-(methylsulfanyl)propyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(1H-imidazol-2-yl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
5-(2-methanesulfonylethyl)-1-phenyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazole
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
N,N-bis(prop-2-en-1-yl)-2-{3',5',6',7'-tetrahydrospiro[cyclohexane-1,4'-imidazo[4,5-c]pyridine]-5'-yl}acetamide
(4aS,7aR)-1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-2-[(3-methylpiperidin-3-yl)methoxy]pyridine
9-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-6-oxa-9-azaspiro[4.5]decane
5-chloro-2-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
2-amino-6-(3,5-difluorophenyl)-4-[3-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
3-methyl-1-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2-chloro-4-fluorophenyl)methyl]-1-cyclopentanecarbonylpiperidine-4-carboxamide
2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-3-ol
2-[(1-benzyl-1H-imidazol-2-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-4-yl)ethyl]amine
3-methoxy-N-{3-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}benzamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
(2S)-2-[5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol
methyl (2S,4S)-1-methyl-4-(2-methyl-1-phenyl-1H-1,3-benzodiazole-5-amido)pyrrolidine-2-carboxylate
N-[3-(3-methoxyphenyl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
1-(4-fluoro-3-methylbenzoyl)-4-(2-methylphenyl)-1,4-diazepane
(1R,2R,6S,7S)-4-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-[1-ethyl-8-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-({5-[(2,6-difluoro-3-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1-methyl-1H-indole-3-carbonyl)pyrrolidin-3-yl]methanol
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
2-methyl-N-[3-(4-methylpiperazin-1-yl)butyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-(azocan-1-yl)-N-[1-(methoxymethyl)cyclopentyl]propanamide