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5-(5-ethylfuran-2-yl)-4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-imidazole
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
methyl 2-[2-(4-fluorophenyl)piperidin-1-yl]acetate
N-[1-(2-methoxyethyl)-7-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
1-(3-fluorobenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(8-{[3-(furan-2-yl)phenyl]methyl}-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
dimethyl({4-[1-(2-methylfuran-3-carbonyl)piperidin-2-yl]phenyl}methyl)amine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(piperidin-4-ylmethyl)benzamide
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]methyl}-2-(methylamino)benzamide
N-cyclopentyl-2-[4-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)morpholin-3-yl]acetamide
N,5,7-trimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-cyclohexyl-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
2-(2-methylphenyl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
2-{1-[6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]-N-methylformamido}acetamide
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl][(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amine
7-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 3-cyclohexyl-2-oxo-1-(1,3-thiazol-2-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
2-ethyl-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrimidine-5-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]acetamide
6-methyl-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,3-benzothiazole
5-chloro-N-[2-(dimethylamino)ethyl]-N-(thiophen-3-ylmethyl)thiophene-2-carboxamide
(3aS,6aR)-5-acetyl-3-[(3,4-dimethoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-methoxy-N-(oxolan-2-ylmethyl)benzamide
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
5-phenyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
6-ethyl-2-(morpholin-4-yl)-N-[1-(pyridin-2-yl)propyl]pyrimidin-4-amine
{3-ethyl-1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}methanol
4-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}benzoic acid
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
1-[3-({[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)piperidin-1-yl]ethan-1-one
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)propanamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(2-methoxyethyl)pyrimidin-2-amine
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[(2-methylpyrimidin-5-yl)methyl]amine
2,5-dimethyl-N-[3-(morpholin-4-yl)propyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-(2,2-difluoroethyl)-2-(dimethylamino)-2-(4-methylphenyl)acetamide
(1S,5R)-N-(4-fluorophenyl)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3R,4S)-4-(5-methylfuran-2-yl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-amine
1-[1-(2-hydroxyacetyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
ethyl 1-[(2-hydroxy-3-methoxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
ethyl 1-{[2-(pyridin-2-yl)pyrrolidin-1-yl]sulfonyl}piperidine-4-carboxylate
9-methoxy-7-(5-methylthiophen-2-yl)-4-(1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,4R)-3-hydroxy-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-4-yl]pyridine-2-carboxamide
4-[4-(4-fluorophenyl)piperazin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{4-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
1-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-3-(furan-2-ylmethyl)urea
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)quinoline