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N-ethyl-2-{[5-(2-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
1,3-dimethyl-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(2,5-dimethylphenyl)ethan-1-one
N-{1-[1-(4-chloro-2-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
3-{6-amino-5-cyano-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]pyridin-2-yl}-1H-pyrazole-5-carboxylic acid
N,5-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(2-{[1-(dimethyl-1,3-thiazol-4-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({methyl[(4-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
(4aS,8aS)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-decahydroisoquinolin-4a-ol
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)piperidine
(3S,7S)-5-(5,6-dimethylpyridine-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-5,6-dimethylpyrimidin-4-amine
2-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}phenyl)ethan-1-ol
5-ethyl-N-(1-methoxybutan-2-yl)-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
8-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.5]decane
1-benzyl-4-oxo-N-(propan-2-yl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
3-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}sulfonyl)pyridine
N-(1H-1,3-benzodiazol-2-yl)-2-{methyl[2-(1H-pyrazol-4-yl)ethyl]amino}acetamide
1-[(4-fluorophenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
5-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-3-ethyl-1,2-oxazole
4-[(5-{imidazo[2,1-b][1,3]thiazol-6-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-propylpiperidine
1-[4-(1H-imidazol-1-ylmethyl)phenyl]-2-(propan-2-yl)-1H-imidazole
5-(quinolin-8-yl)pyrazin-2-amine
1-(3-chlorophenyl)-4-(3-hydroxy-4-methylbenzoyl)-5-methylpiperazin-2-one
(1R,2R,4R)-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-{3-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]propanamido}benzamide
2-(2H-indazol-2-yl)-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}ethan-1-one
(2S,4S)-4-amino-1-(5-chloropyridine-2-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
5-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}isoquinoline
4-(quinolin-8-yl)thiophene-2-carboxylic acid
N-{[(2S,4S)-4-fluoro-1-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]pyrrolidin-2-yl]methyl}piperidine-1-carboxamide
[(3-cyclopropyl-1H-pyrazol-5-yl)methyl](methyl)(oxan-2-ylmethyl)amine
1-benzyl-5-[(1-benzylpiperidin-4-yl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(3-chlorophenyl)methyl][(1,4-dimethyl-1H-pyrazol-5-yl)methyl]methylamine
1-[(3,5-dimethylphenyl)methyl]-4-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]piperazin-2-one
N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
2,5-dimethyl-N-[2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-1,3-thiazole-4-carboxamide
2-amino-6,7-dimethoxy-4-(piperidin-3-yl)-5H-indeno[1,2-b]pyridine-3-carbonitrile
4-ethoxy-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidin-2-amine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
8-[(4-fluoro-3-methylphenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[5-chloro-2-(propan-2-yloxy)phenyl]-2-(4-hydroxypiperidin-1-yl)acetic acid
2-{1-cyclopentyl-4-[(2,3-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(4-hydroxyphenyl)methyl]-2-(propan-2-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
4-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-1-cyclopentylpiperazin-2-one
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
4-(4-hydroxy-4-phenylpiperidine-1-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one