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{3-[(4-fluorophenyl)methyl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl}methanol
N-(3-methylbutyl)-3-[(2-oxopiperidin-3-yl)sulfamoyl]benzamide
2-(3-chloro-4-methoxyphenyl)-5,6-dimethylpyridine-3-carboxamide
6-{2-[ethyl(methyl)amino]butyl}-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2,6-dimethylpyrimidine-4-carboxamide
6-(methoxymethyl)-1-methyl-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{1-[3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carbonyl]cyclopropyl}methanol
3-methyl-N-({3-methyl-7-[2-(trifluoromethyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
3-{5-[(3-hydroxy-4-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-(4-chlorophenyl)-2-({6-methylimidazo[1,2-a]pyridin-2-yl}formamido)acetic acid
2-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]phenol
5-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
4-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}benzene-1-sulfonamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(pyridin-4-ylsulfanyl)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-[2-(pyridin-4-ylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
1-{4-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]piperidin-1-yl}butan-1-one
1-ethyl-4-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}piperazin-2-one
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-4-(trifluoromethyl)pyrimidin-2-amine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-tert-butyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-hydroxypyrimidine-5-carboxamide
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
1-[(2,3-difluorophenyl)methyl]-N-phenylpiperidin-3-amine
2-{[(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)oxy]methyl}pyridine
(3S,4S)-1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
(3-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}phenyl)methanol
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
3-(5-methyl-4H-1,2,4-triazol-3-yl)-1-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]urea
N-(1-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
1-{1-[4-(5-phenylpentanamido)phenyl]piperidin-4-yl}piperidine-3-carboxamide
(4aS,7aR)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[(1-cyclohexanecarbonylpiperidin-3-yl)methyl]naphthalene-1-carboxamide
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2,8-dimethylquinoline
3-methyl-N-[6-methyl-4-(1-methyl-1H-pyrazol-4-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]benzamide
(3R,4R)-1-(3-fluoro-4-methylbenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
2-(methylamino)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3-thiazole-4-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-(3,4-difluorophenyl)acetamide
2-(1H-indol-3-yl)-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide
1-(3-chlorophenyl)-4-[3-(pyrrolidin-1-yl)piperidin-1-yl]piperidine
2-[3-(8-methoxyquinolin-5-yl)phenoxy]propanamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[4-(pyrrolidin-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
4-[4-(2H-1,3-benzodioxol-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-(2-fluorophenyl)piperidin-4-ol
1-{4-[(dimethylsulfamoyl)amino]phenyl}-N-(thiophen-3-ylmethyl)piperidin-4-amine
3-({[1-(2-phenylethyl)piperidin-4-yl]oxy}methyl)pyridine
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2-(4-fluorophenyl)piperidine
1-{4-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]piperidin-1-yl}ethan-1-one
5-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}thiophene-2-carboxylic acid