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N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-(methoxymethyl)-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-{8-[1-(methylsulfanyl)propan-2-yl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
1-cycloheptyl-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(1H-pyrazol-1-yl)benzamide
{5-methyl-7-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
4-[(1R,7S)-3-(3,4-dimethylphenyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-3-phenylpyrrolidin-3-ol
3-cyclopentyl-6-(oxolan-3-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
(1S,5R)-6-benzoyl-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclohexyl-3-(2-{methyl[2-(pyridin-2-yl)ethyl]carbamoyl}ethyl)piperidine-1-carboxamide
ethyl 1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
1-(piperidin-3-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(1-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}propyl)piperidine-1-carboxamide
N-[(3S,4R)-4-propyl-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidin-3-yl]methanesulfonamide
5,6-dimethyl-N-(oxan-4-yl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N,N-dimethyl-3-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]propanamide
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)-4-(piperidin-1-yl)piperidine
N3-methyl-N5-[(2-methylphenyl)methyl]-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-benzyl-N-(cyclopropylmethyl)-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
8-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-2-methyl-2,8-diazaspiro[4.5]decan-3-one
1-{1-[(2,6-dimethylphenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrimidin-2-amine
[1-(2-methylpyrimidin-4-yl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
2-[(2-cyclopentylacetamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
6-chloro-2-methyl-4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}quinoline
1-ethyl-3-methyl-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}-1H-pyrazole-5-carboxamide
N-(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
8-{[3-(thiomorpholine-4-carbonyl)-1,2-oxazol-5-yl]methoxy}quinoline
9-ethyl-3-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}-9H-carbazole
3-(3-fluorophenyl)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
4-methoxy-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine
2-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-N-(5-methyl-1,2-oxazol-3-yl)-2-oxoacetamide
[1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidin-2-yl]methanol
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
5-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
8-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,2,3-thiadiazole-5-carboxamide
7-fluoro-3-methyl-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
1-{2-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[3-(dimethylamino)propyl]-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
5-methyl-4-{[1-(1,3-thiazol-2-yl)ethyl]amino}-N-[2-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
5-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-1H-indole-2-carboxamide
2-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
1-[(4aS,8aS)-4a-hydroxy-7-(pyridin-4-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-3-methylbut-2-en-1-one
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
N-[1-(1,1-dioxo-1λ6-thian-4-yl)piperidin-4-yl]-1H-pyrazole-4-carboxamide