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methyl 2-{2-oxo-4-[(3-phenyl-1,2,4-thiadiazol-5-yl)carbamoyl]piperazin-1-yl}acetate
2-[(3-methoxyphenyl)methyl]-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3,3-dimethyl-1-(9-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3,9-diazaspiro[5.5]undecan-3-yl)butan-1-one
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxylate
1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-4-methylpiperazine
4-(5-ethyl-1,3-oxazole-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrrole
(1R,5R)-6-(1-benzofuran-2-ylmethyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(3-hydroxypropyl)acetamide
(2S,4S)-4-{[(3-fluorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
2-{2-[4-(1H-pyrazol-3-yl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-1-yl}acetic acid
3-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-6-(1-methyl-1H-imidazol-2-yl)pyridazine
4-(oxolan-3-yl)-1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazole
2-methyl-5-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]aniline
5-[(6-chloro-2H-chromen-3-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-({2-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[1-(azepane-4-carbonyl)piperidin-4-yl]-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)-6-methylpyridazine
7-fluoro-2-methyl-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine-1-carbonyl]quinoline
4-(4-{[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
2-amino-3-ethyl-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-acetamido-N-(4-pentylphenyl)pyrrolidine-1-carboxamide
4-propyl-1-[4-(trifluoromethyl)benzoyl]-1,4-diazepan-5-one
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-methyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
2-oxo-4-phenyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butanamide
2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyridin-4-yl)ethan-1-ol
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]benzamide
1-[(3-methylpyridin-2-yl)methyl]-4-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-{3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-oxopropyl}piperidin-2-one
ethyl 1-[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-2-carboxylate
2-(4-methoxypyrimidin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-propyl-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]-2-methylphenol
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(2-methyloxane-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{2-carbamoyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidine-1-carboxamide
3-benzyl-4-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}piperazin-2-one
7-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[2-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-{3-[3-(3,4-difluorophenyl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
3-[2-(2,4-difluorophenyl)ethyl]-1-(1,3-thiazole-4-carbonyl)piperidine
(3aS,6aS)-2-[(4-butylphenyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
1-{2-hydroxy-3-[4-methoxy-2-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
1'-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
methyl({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine