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{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-(piperidin-4-ylmethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
[5-({1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyridin-2-ylmethyl})amine
N-cyclopropyl-2-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]pyridine-4-carboxamide
4-[(dimethylamino)methyl]-4-hydroxy-N-(3-methoxyphenyl)azepane-1-carboxamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N'-(adamantan-1-yl)-N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]propanediamide
(1S,5R)-3-(2-methylfuran-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[(5-methylthiophen-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-[1-(5-hydroxypyrazine-2-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetamide
methyl 2-{[(3S,4R)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylate
4-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-3,3-dimethylpiperazin-2-one
4-{[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl}thiomorpholine
5-(3-fluoro-5-methylphenyl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
2-(3-chlorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
N-(2-{4-[(2-phenyl-1,3-oxazol-4-yl)methyl]morpholin-2-yl}ethyl)acetamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]amine
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-propyl-1,3,4-oxadiazole-2-carboxamide
(3S,4R)-1-[(2,4-difluorophenyl)methyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
4-(cyclopentylamino)-1-(2-phenylethyl)pyrrolidin-2-one
N-{3-[(2-ethylphenyl)carbamoyl]phenyl}-6-oxo-1-propylpiperidine-3-carboxamide
1-(cyclohexylmethyl)-6-oxo-N-(3-phenylpropyl)piperidine-3-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
8-chloro-2-({[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]amino}methyl)quinolin-4-ol
2-({4-[4-(3-propoxypiperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
N,3,5,7-tetramethyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H-indole-2-carboxamide
2-methyl-6-{1-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
(3R,5S)-N-[3-(furan-2-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-{[2-({[1-(2-methoxyethyl)piperidin-3-yl]methyl}(methyl)carbamoyl)phenyl]amino}acetic acid
2-methyl-3-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
4-(3,4-dichlorophenyl)-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-1-(pyridin-2-ylmethyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-(4-{[4-methoxy-3-({1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}piperazin-1-yl)ethan-1-one
1-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-5-oxopyrrolidine-3-carboxylic acid
1-[(2-fluorophenyl)methyl]-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazin-2-one
6-tert-butyl-N-[1-(furan-2-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[(3S,5R)-1-(6-cyclopropylpyrimidin-4-yl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(3-ethoxypropyl)-2-methylimidazo[1,2-a]pyridine-6-carboxamide
5-[1-(but-2-ynoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
6-fluoro-4-hydroxy-N-methyl-N-[2-(morpholin-4-yl)propyl]quinoline-3-carboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-(2-phenoxyethyl)-1H-pyrazole-3-carboxamide
4-(4-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol