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N-butyl-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(furan-2-ylmethyl)-3-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}piperidine
N-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)propanamide
4-{6-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
3-(3-chlorobenzoyl)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine
2-{5-[1-(4-methylpiperidin-1-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
4-benzyl-3-ethyl-1-[6-(methoxymethyl)pyrimidin-4-yl]-1,4-diazepan-5-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-1H-pyrazole-4-carboxamide
2,6-dimethoxy-3-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}pyridine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidine
1-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
2-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]phenoxy}ethan-1-ol
3-(2-amino-1,3-thiazol-4-yl)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
5-(2-fluorophenoxymethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-[(4-methanesulfonylphenyl)methyl]-3,9-diazaspiro[5.5]undecane
8-(3-methoxybenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-[3-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
5-(4-methyl-1,3-oxazol-5-yl)-3-(1-phenylcyclopropyl)-1-propyl-1H-1,2,4-triazole
3-[(3R,4S)-1-[(3-chloro-4-fluorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
2-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]benzoic acid
N'-cyclopentyl-N-{3-[ethyl(methyl)amino]-2-methylpropyl}butanediamide
4-{2-[2-(1-benzofuran-5-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
N-cycloheptyl-4-oxo-1-(propan-2-yl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
4-[(2-cyclopentyl-1H-imidazol-1-yl)methyl]-1H-indole
4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-N-[2-(propan-2-ylsulfanyl)ethyl]benzene-1-sulfonamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2-hydroxy-3-methoxybenzamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(methylamino)-1,3-thiazole-4-carboxamide
1-{2-oxo-2-[(3S,4R)-3-propyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]ethyl}azepan-2-one
2-acetyl-8-(6-chloroquinolin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
{5-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]furan-2-yl}methanol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(dimethylamino)-N-methyl-2-(4-methylphenyl)acetamide
4-[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)amino]pyrimidine-5-carboxylic acid
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propan-1-one
2-{imidazo[1,2-a]pyridin-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(adamantan-1-ylsulfanyl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
3-{4-[(5-phenylthiophen-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-amine
1-cycloheptyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(3S,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3-ethyl-1H-pyrazole-5-carboxamide
5-{[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-(3-ethoxypropyl)-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-[(4-methylphenyl)amino]-N-(pyridin-2-ylmethyl)cyclopentane-1-carboxamide
N-ethyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
ethyl 4-benzyl-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidine-4-carboxylate
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-[(3R,4S)-4-(dimethylamino)-1-[(2-phenylphenyl)methyl]piperidin-3-yl]propan-1-ol
2-butoxy-1-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one