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3-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]methyl}-7-fluoro-1-(2-phenylethyl)-1,2-dihydroquinolin-2-one
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-(pyridin-2-ylmethyl)pyrrolidin-3-amine
1-[3-(4-methylpiperazine-1-carbonyl)phenyl]-3-[4-(1H-pyrazol-1-yl)butan-2-yl]urea
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(pyrazin-2-yl)-1,4-diazepan-6-ol
6-fluoro-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-(1H-imidazol-2-ylmethyl)-2-[(3-methoxyphenyl)methyl]morpholine
2-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]pyridine-3-carbonitrile
3-(4-chlorophenyl)-5-[(1R,2R)-2-phenylcyclopropanecarbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-(morpholin-4-yl)-2-(pyridin-3-yl)-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethan-1-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-[(4-methoxyphenyl)methyl]-6-[3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1,3-benzoxazole
N-[3-(azepan-1-yl)-2-hydroxypropyl]-4-chloro-1-methyl-1H-pyrazole-5-carboxamide
3-[(3R,4R)-4-amino-3-hydroxypiperidine-1-carbonyl]-6-fluoro-7-(morpholin-4-yl)-1,4-dihydroquinolin-4-one
9-(2-hydroxyethyl)-1-methyl-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[2-(2-fluorophenyl)ethyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
(3S,4R)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
9-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[(4,4-difluoropiperidin-1-yl)methyl]-8-methylquinoline
1-cyclopentyl-4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]pyrrolidin-2-one
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-2-(4-fluorophenyl)piperidine
N-(butan-2-yl)-2,4-dimethoxy-N-(thiophen-3-ylmethyl)benzamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl]propanamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-3,4,5-trimethoxy-N-(oxolan-2-ylmethyl)benzamide
1-[4-(quinazolin-4-yl)piperazin-1-yl]-3-(thiophen-3-yl)propan-1-one
4-(3-chlorophenyl)-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-[(adamantan-1-ylformamido)methyl]-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
(3aS,6aS)-2-cyclobutanecarbonyl-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-5-[4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
[(3R,4R)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N4,N4,5-trimethyl-N2-[4-(1H-pyrazol-1-yl)butan-2-yl]pyrimidine-2,4-diamine
1-[(8-methoxyquinolin-2-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-[1-(9H-purin-6-yl)piperidin-4-yl]propan-2-ol
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethylquinoxaline-5-carboxamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-cyclopentyl-3-[5-(1H-pyrrole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-2-(naphthalen-1-ylmethyl)morpholine
4-(4-chloro-2-hydroxybenzoyl)-1-[(2-fluorophenyl)methyl]piperazin-2-one
N-{[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]methyl}-1H-indazole-3-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
4-{3-[2-(furan-3-yl)-1H-imidazol-1-yl]phenyl}-1,3-thiazole
2-(4-methoxyphenyl)-5-[(3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
2-({[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(methyl)amino)propanamide
2-{[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]amino}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide