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4,6-dimethoxy-2-[3-(pyridin-3-yl)propyl]pyrimidine
N-[3-(methylsulfanyl)propyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-(4-methyl-1,4-diazepane-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(4-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-[4-methyl-3-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
1-{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}-2-methyl-1,4-diazepan-5-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
5-cyclopropanecarbonyl-1'-(thiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
2-(5-fluoro-2-methoxyphenyl)-2-[methyl(1H-pyrazol-5-ylmethyl)amino]acetic acid
4-(7-chloroquinolin-4-yl)-2-[(4-methylpiperidin-1-yl)methyl]phenol
2-[(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propan-1-ol
(4aS,7aR)-1-[2-(4-fluoro-3-methylphenyl)acetyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
2-[5-(1-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
4-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidine
N,2-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-benzofuran-7-carboxamide
5-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-2-fluorobenzamide
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,2-dimethyl-1H-1,3-benzodiazole-5-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-8-fluoroquinoline-2-carboxamide
N-(2-chloro-5-methylphenyl)-3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
(3aR,6aS)-5-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-{[3-(trifluoromethoxy)phenyl]methyl}urea
2,5-dimethyl-3-[4-(1,3-thiazol-4-ylmethyl)piperazin-1-yl]pyrazine
3-[(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)oxy]pyridine
1-(3-chloro-5-fluorobenzoyl)-3-(3-methoxypropyl)piperidine
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-methylbut-2-en-1-one
N-[2-(1,3-benzothiazol-2-yl)ethyl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
methyl 1-(3-{4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
3-methoxy-1-[3-(2-phenylethyl)piperidin-1-yl]propan-1-one
N-[2-(3-fluorophenyl)-2-hydroxyethyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)-3-(1H-pyrazol-5-yl)piperidine
6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
N-(2-methylpropyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-ethyl-N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
methyl({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
2-(2-hydroxypropyl)-9-(1,3-thiazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methoxyethyl)-8-(1-methoxypropan-2-yl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-propylbutanamide
(2S,4S)-4-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamido]-N-ethyl-1-(pent-2-yn-1-yl)pyrrolidine-2-carboxamide
3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-1-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
{5-[({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)methyl]furan-2-yl}methanol
(1-{[methyl({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}cyclobutyl)methanol
2-(3-fluorophenyl)-N-[3-(1H-pyrazol-1-yl)propyl]-1,3-benzoxazole-5-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-7-methanesulfonyl-N,4-dimethylquinazolin-2-amine
2-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
methyl 7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-3-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{4-[3-(dimethylcarbamoyl)pyridin-2-yl]phenoxy}acetic acid