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N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-(adamantan-2-ylmethyl)-6-{[benzyl(ethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[4-(morpholin-4-ylmethyl)phenyl]-3-propoxypiperidine-1-carboxamide
4-cyclopentanecarbonyl-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(4-chloro-2-methylbenzoyl)-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine
3-(4-methoxy-2-methylbenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-fluorophenyl)methyl]piperidin-3-ol
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-N-(pyridin-2-ylmethyl)aniline
(3R,4R)-4-ethyl-1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperidine-3,4-diol
2-{1-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidin-3-yl}benzoic acid
N-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
5-ethyl-1-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-4-phenyl-1H-imidazole
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[3-(pyrrolidin-1-yl)propyl]amine
1-cyclopentyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(2-methylphenyl)methyl]amine
5-{[3-(4-tert-butylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-ethyl-1H-1,2,4-triazole
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-{[(5-methyl-1,3,4-oxadiazol-2-yl)amino]methyl}pyrrolidin-2-yl]methanol
(4aS,7aR)-1-[(4-fluoro-3-methylphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-1-(1-benzofuran-2-ylmethyl)-4-methylpiperidine-3,4-diol
5-[4-(2-methoxyphenyl)piperazin-1-yl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
6-fluoro-4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-[2-(dimethylamino)ethyl]-3-methyl-N-[(5-methylthiophen-2-yl)methyl]furan-2-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}propanamide
9-[2-(3-fluorophenyl)ethyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1H-1,3-benzodiazol-2-ylmethyl)({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
(1R,7S)-3-(2-ethoxyethyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
(1R,3S,5S)-8-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-8-azabicyclo[3.2.1]octan-3-ol
2-benzyl-8-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecane
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2-(thiophen-3-yl)acetamide
(2R)-2-amino-1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-3-phenylpropan-1-one
5-(dimethylamino)-2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dihydropyridazin-3-one
1-[3-(benzyloxy)propyl]imidazolidin-2-one
2,2-diethyl-4-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]morpholine
methyl 6-{[butyl(methyl)amino]methyl}-3-(2-fluorobenzamido)thieno[2,3-b]pyridine-2-carboxylate
5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(2-fluorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazole
2-[(2-methoxyethyl)(methyl)amino]-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
2-(4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrrolidine-1-carboxamide
1-(cyclopropylmethyl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazine
2-ethyl-1-[(4-methoxyphenyl)methyl]-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1,4-dihydropyridin-4-one
1-(2-methoxyethyl)-N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)pyrrolidine-3-carboxamide
2-(5-acetylthiophen-3-yl)-N-(thiophen-3-ylmethyl)acetamide
3-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanoic acid
(4aR,7aS)-1-methyl-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione