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1-methyl-1'-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
5-{[methyl({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]methyl}pyrimidin-2-amine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-pyrrol-1-yl)propan-1-one
1-(4-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)-1H-1,2,4-triazole
(1R,5R)-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1r,4r)-4-[({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]cyclohexan-1-ol
N-cyclopentyl-5-phenyl-N-(thiophen-3-ylmethyl)-1,2-oxazole-3-carboxamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
(4S)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3,3,4-trimethylpiperidin-4-ol
2-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(2-methylphenoxy)piperidine
5-methoxy-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}furan-2-carboxamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
6-[2-(4-fluorophenyl)-3-oxopiperazine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(4-chlorophenyl)ethyl]propanamide
N-(2-methoxyethyl)-1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
7-methoxy-3-{[4-(pyridin-4-ylmethyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5-phenyl-1,2,4-oxadiazol-3-amine
9-(4-fluoro-3-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-chlorophenyl)methyl]-8-[(2S)-3-hydroxy-2-(methylamino)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
3-[5-(pyridin-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-(3-methyl-1H-pyrazol-1-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(morpholin-4-yl)propan-1-one
methyl (2S)-2-[(5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidin-6-yl)formamido]-3-phenylpropanoate
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(4,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methylacetamide
(3S,4R)-1-(1,4-dithiepan-6-yl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
methyl 4-({3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}methyl)benzoate
(3aS,6aR)-5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1S,5R)-3-(2-cyclopentylacetyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(1-{[1-(1,4-dimethylpiperidine-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
2-ethyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]pyrimidine-5-carboxamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
3-(4-chloro-2-ethylphenyl)-1-{3-[(1-methylpiperidin-4-yl)oxy]propyl}urea
3-(pyridin-3-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-[4-(methylsulfanyl)phenyl]-2-(morpholin-4-yl)acetic acid
5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
3-{3-[1-(dimethylamino)ethyl]phenyl}-5,6-dimethyl-1,2-dihydropyridin-2-one
1-(cyclopropylmethyl)-5-(4-ethyl-5-methylthiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
8-{[4-(diethylamino)-2-methylphenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
3-{4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyridine
1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
[2-ethoxy-5-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenyl]methanol