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1-{2-[(2,3-dimethoxyphenyl)formamido]ethyl}-N-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
9-[(3-chloro-1H-indol-2-yl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-({1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
2-(5-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
4-methyl-6-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]pyrimidin-2-amine
3-{2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-{3-[(1R,9S)-5-amino-4-cyano-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-trien-3-yl]phenoxy}acetamide
3-ethoxy-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]benzamide
N-cyclohexyl-3-[2-(dimethylamino)-2-(2-methylphenyl)acetamido]propanamide
[(3R,4R)-1-(2-cyclopropylpyrimidine-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methylpiperidine-3-carboxamide
3-[(2,4-difluorophenyl)methyl]-1-(6-methylpyridazin-3-yl)piperidine-3-carboxylic acid
N-(furan-3-ylmethyl)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
1-methyl-N-[3-(phenylsulfanyl)propyl]piperidine-2-carboxamide
1-methyl-2-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1H-indole
N-({5-[3-(dimethylamino)-2,2-dimethylpropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
(1S,5R)-N,N-dimethyl-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}[(1-methyl-1H-pyrazol-5-yl)methyl]amine
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
2-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
6-[(3-hydroxy-3-methylbutyl)(methyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-4H-1,2,4-triazole
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-(thiolan-3-yl)piperidine
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-4-methylpyrimidine-5-carboxamide
5-methoxy-2-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)pyridin-4-ol
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
3-[2-(2,3,6-trimethylphenoxy)acetamido]butanoic acid
(4aR,8aR)-2-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]propanoate
1-methyl-N-{1-oxaspiro[4.5]decan-3-yl}-1H-indole-6-carboxamide
[(3R,4R)-1-[3-(dimethylamino)pyrazin-2-yl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
2-(2-fluoro-3-methylphenyl)-N,N-dimethylpyridine-3-carboxamide
[5-({ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)furan-2-yl]methanol
1-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(1-benzofuran-2-yl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-methylpiperazine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-(4-chlorophenoxy)-1-{4-[2-(methoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethan-1-one
4-(2-hydroxypyridine-3-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 4-({2-[(thiophen-2-ylmethyl)carbamoyl]ethyl}amino)piperidine-1-carboxylate
3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-5-chloro-1,2-dihydropyridin-2-one
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-5-methyl-1,2-oxazole
methyl 4-{3-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]propanamido}benzoate
1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(pyrazin-2-yl)propan-1-one
N-ethyl-4-hydroxy-N-(2-methoxyethyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2,2-dimethyl-N-(1-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
4-(4-chlorophenyl)-3-(1-ethyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one