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2-methoxy-5-{2-[5-(1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}phenol
(3S,4S)-1-(2,6-dimethylquinoline-3-carbonyl)-4-(propan-2-yloxy)pyrrolidin-3-ol
3-[4-(benzyloxy)piperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2-(azepan-1-yl)-2-(2,4-dimethoxyphenyl)acetic acid
2-methoxy-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
1-methyl-4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperazine
N-(1-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
4-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(3-fluoro-4-phenylbenzoyl)piperidine
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(3,4-difluorophenyl)-N-[2-(pyrazin-2-yl)ethyl]propanamide
3-(6-cyanopyridin-3-yl)-1-cyclohexyl-1-(pyridin-2-ylmethyl)urea
N-[2-(morpholin-4-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-(3-ethyl-1,2-oxazole-5-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
5-(cyclobutylmethyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-[2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
3,5-dichloro-4-methyl-N-[2-(N-methylmethanesulfonamido)ethyl]benzamide
1-(1-benzoxepine-4-carbonyl)-4-methyl-1,4-diazepan-6-ol
4-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)piperazine-1-carboxamide
5-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]pyrazin-2-ol
5-methoxy-1-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-indole-2-carboxamide
N4-[(3-fluoro-4-methylphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
methyl 5-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-5-oxopentanoate
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(1-benzothiophen-5-ylmethyl)acetamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}pyrazin-2-amine
2-(methylsulfanyl)-N-[(2R,3R)-2-(prop-2-en-1-yloxy)-1'-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}pyrimidin-2-amine
3-phenyl-1-{1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-4-yl}propan-1-ol
3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-(4-methanesulfonylphenyl)urea
1-(3-{2-azaspiro[4.4]nonan-2-ylmethyl}phenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-[2-(3-methoxyphenyl)ethyl]-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
methyl 4-{[4-(benzyloxy)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
8-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
8-[(4-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(4-chlorophenyl)cyclopropyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propan-1-one
N-(5-pentyl-1,3,4-thiadiazol-2-yl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carboxamide
4-(2-fluoro-4-methoxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{1-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-ethylpentanamide
4-(2-chloro-6-fluorobenzoyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]propan-1-ol
1-[(4-fluorophenyl)methyl]-3-{2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-(2-{[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}ethyl)-1,3-oxazolidin-2-one
N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[3-(methylamino)propyl]-4-(piperidin-3-yl)benzamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(methylsulfanyl)pyrimidine-5-carboxamide