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3-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)benzoic acid
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
15-methyl-13-oxo-N-[2-(pyridin-4-yl)ethyl]-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
N-(2-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
4-methyl-3-phenyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-pyrazole-5-carboxamide
7-fluoro-N,3-dimethyl-N-[4-(morpholin-4-yl)butyl]-1-benzofuran-2-carboxamide
N-(1-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylcyclopropanecarboxamide
1-{3-[4-(azepan-1-ylmethyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N-cyclopentyl-N'-[2-(quinolin-8-yloxy)ethyl]butanediamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
3-({1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)pyridine
5-[(2,4-dimethoxyphenyl)methyl]-8-methoxy-2-[3-(trifluoromethyl)phenyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-(2-methoxyethyl)-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
8-{3-[5-(4-methylphenyl)furan-2-yl]propanoyl}-2,8-diazaspiro[4.5]decan-3-one
1-{2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
ethyl 4-(2-amino-1,3-benzothiazole-5-carbonyl)piperazine-1-carboxylate
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,4-difluorobenzamide
2-butyl-4-methyl-N-[2-(methylsulfanyl)phenyl]-3-oxopiperazine-1-carboxamide
N-methyl-2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,1,3,6-tetramethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
1-(2,6-dimethylhept-5-en-1-yl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-(tert-butylsulfamoyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
1-methyl-4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
2,2-difluoro-N-[2-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)ethyl]acetamide
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]pyridin-2-amine
N-cyclohexyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
3-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,5-dimethyl-2-(2-methylpropanamido)benzamide
3,3-dimethyl-1-{2-oxo-2-[2-(2-phenylethyl)piperidin-1-yl]ethyl}urea
N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
N,N-dimethyl-3-{1-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]piperidin-3-yl}propanamide
2-[(1,3-benzothiazol-2-yl)amino]-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
4-methoxy-N-(2-methoxyethyl)-2-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
1-(4-methyl-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrimidin-5-yl)ethan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-phenylpropyl)benzamide
3-cyclohexyl-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
5-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-phenyl-1H-1,2,4-triazole
N-{2-[methyl(phenyl)amino]ethyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-(3-chlorophenyl)-4-(piperidin-3-yl)piperazine
2-[5-(methoxymethyl)-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
N-({3-methyl-7-[3-(2-oxopyrrolidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
N-(1-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
3-(3-fluorophenyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(pyrrolidin-3-yl)-N-(quinolin-5-yl)benzamide
5-[1-(4-chlorobenzoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyridine-3-carbonitrile
ethyl 4-{2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetyl}piperazine-1-carboxylate