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N-[2-(4-ethylmorpholin-2-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-butyl-1-methyl-4-(5-propylthiophene-3-carbonyl)piperazin-2-one
(1S,5R)-3-(2,5-dimethylfuran-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-[1-(pyridin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
1-[(4-methylphenyl)methyl]-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
2-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1-methylpiperidin-4-amine
2-(3-methyl-1,2-oxazol-5-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
1-methyl-4-{[5-(5-phenyl-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}-4-methylbenzamide
6-ethyl-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidin-4-amine
1,7-dimethyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,4-dioxo-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-5-carboxamide
N-cyclopropyl-3-[5-(3-phenylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
(4aS,7aR)-1-(6-aminopyridine-3-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(2S)-2-aminopentanoyl]-N-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}[(2-methoxynaphthalen-1-yl)methyl]methylamine
7-[2-(1H-imidazol-1-yl)propanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-fluorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N'1-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropane-1,1-dicarboxamide
7-fluoro-3-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)-3,4-dihydroquinazolin-4-one
N-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1-(pyridin-3-ylmethyl)piperidin-4-amine
3-(4-fluorophenyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
3-{[(cyclohexylmethyl)amino]methyl}-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-(3-chloro-4-methoxyphenyl)-5-oxo-N-[2-(pyrazin-2-yl)ethyl]pyrrolidine-3-carboxamide
3-methoxy-2-(2,4,6-trimethylphenyl)pyridine
methyl 3-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}benzoate
N-[3-({[(4-methoxynaphthalen-1-yl)methyl]amino}methyl)-5-(4-methylpiperazine-1-carbonyl)phenyl]acetamide
2-(2,4-dichlorophenoxy)-N-methyl-N-[3-(oxolan-2-yl)propyl]acetamide
(3S)-3-ethyl-4-[(4-methoxypiperidin-1-yl)sulfonyl]morpholine
1-[4-(2-methylphenoxy)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
2-[4-(3-phenoxyphenyl)-1H-1,2,3-triazol-1-yl]propanoic acid
2-{4-[3-(1H-imidazol-2-yl)benzoyl]piperazin-1-yl}pyrimidine
2-ethyl-8-(5-propyl-1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)[2-methyl-2-(morpholin-4-yl)propyl]amine
1-(3-methylbut-2-en-1-yl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-cyclohexyl-3-[2-(dimethylamino)-2-(3-methylphenyl)acetamido]propanamide
3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
2-(3-methylbutyl)-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[(2-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-[3-(methylsulfanyl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-{2-[1-(3-methylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}methyl)pyridin-2-amine
9-(2-methoxyethyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-acetylphenoxy)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
ethyl 4-benzyl-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine-4-carboxylate
7-[(2,3-difluorophenyl)methyl]-2-(1H-indole-6-carbonyl)-2,7-diazaspiro[4.5]decane