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3-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
1-{[1-(2-methoxyethyl)-6-methyl-2-oxo-1,2-dihydroquinolin-3-yl]methyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
1-[(4-fluorophenyl)methyl]-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1,4-diazepane
3-(oxolan-2-ylmethyl)-5-[1-(2-phenylacetyl)piperidin-4-yl]-5-(pyridin-2-yl)imidazolidine-2,4-dione
ethyl 1-ethyl-5-(2,3,4,9-tetrahydro-1H-carbazole-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-(2H-1,3-benzodioxol-5-yl)-3-methylpyridin-2-amine
ethyl 2-(1-{2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamido}cyclohexyl)acetate
2-(3,4-difluorophenyl)-5-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-chloro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyridine-3-carboxamide
(4aS,8aR)-N-(dimethyl-1,2-oxazol-4-yl)-1-(3-hydroxypropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
1-[benzyl(methyl)amino]-3-(5-{[bis(2-hydroxyethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
1-cyclopentyl-4-[4-methoxy-2-(3-methoxypyrrolidine-1-carbonyl)phenoxy]piperidine
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-chloro-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N,N-diethyl-1-[(1s,4s)-4-[2-(4-methoxyphenyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(1R,3S)-7-(2,3-dihydro-1H-inden-2-yl)-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
1-(2-hydroxyethyl)-5-{[5-(methoxymethyl)furan-2-yl]methyl}-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[5-oxo-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(pyrazin-2-yl)acetamide
8-(3-aminopropanoyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-(pyridin-4-yl)propyl]-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-4-carboxamide
propyl 4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(2S)-oxolane-2-carbonyl]piperidine-4-carboxylic acid
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
2-methoxy-1-[4-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)piperidin-1-yl]ethan-1-one
6-methyl-2-(2-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)-3,4-dihydropyrimidin-4-one
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
N-[(3S,4R)-4-(propan-2-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanesulfonamide
2-{2-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
1-(4-chlorophenyl)-4-(4-hydroxy-3-methoxybenzoyl)-5-methylpiperazin-2-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methanol
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
N-cyclopropyl-4-methoxy-3-{[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]oxy}benzamide
1-(cyclopropylmethyl)-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]-2-(propan-2-yl)-1,4-diazepane
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1H-pyrazol-1-yl)propan-1-one
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2,4-dimethylpyrimidine-5-carboxamide
3-(oxolan-3-yl)-5-[3-(1H-pyrazol-1-yl)propyl]-1,2,4-oxadiazole
N-[1-(2,5-difluorophenyl)cyclopropyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-[(2-methylphenyl)methoxy]azetidine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
(2S)-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-hydroxy-3-phenylpropanamide
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(2,2,2-trifluoroethyl)-1,3-oxazole-4-carboxamide
3-({[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
(1S,5R)-3-[2-(2,3-difluorophenyl)acetyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(diethylamino)ethyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-({1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]propanamide
4-[2-(4H-1,2,4-triazol-4-yl)ethyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide