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4-({4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}methyl)phenol
1-(furan-2-ylmethyl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
N-(3-aminopropyl)-2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-ethyl-N-(pyridin-4-ylmethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
3-[4-(methylsulfanyl)benzoyl]-1-(3-phenylprop-2-yn-1-yl)piperidine
methyl 3-[(cyclohexylformamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
(3R,4S)-4-(4-methoxyphenyl)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidin-3-amine
N-(1-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
6-[4-(2,1,3-benzothiadiazol-4-ylmethyl)piperazin-1-yl]pyridine-3-carboxamide
(3R,4R)-4-(hydroxymethyl)-1-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)piperidin-3-ol
N-cyclopropyl-1-[1-(pyridazine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-[(3-methoxyphenyl)methyl]-3-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)piperazin-2-one
7-methyl-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
1-benzyl-8-methyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5S)-N-cyclopentyl-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]urea
3-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-amido]pyrrolidine-3-carboxylic acid
1-[3-(furan-2-yl)phenyl]-3-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}urea
2-(5-chloro-2-methoxypyridin-4-yl)-5-fluoro-4-(pyrrolidin-1-yl)pyrimidine
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(propan-2-yl)pyrimidin-4-amine
[3-benzyl-1-(quinolin-8-ylmethyl)piperidin-3-yl]methanol
6-(6-hydroxypyridine-3-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-5-(2-phenylethyl)-1H-imidazole
4-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-3-yl}benzoic acid
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(1,3-thiazol-2-yl)piperidin-4-ol
2-methoxy-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
4-cyclopentyl-2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyrimidine
3-({[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-3-yl]oxy}methyl)pyridine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
2-[(3-methoxyphenyl)methyl]-8-(2-phenylacetyl)-2,8-diazaspiro[4.5]decan-3-one
5-(dimethylamino)-2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,3-dihydropyridazin-3-one
2-(1H-imidazol-2-yl)-N-(2-phenylethyl)benzamide
2-(4-ethylpiperazin-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]-2,3-dihydro-1H-indene-2-carboxamide
N'-(4-methylphenyl)-N-[3-(pyridin-4-yl)propyl]propanediamide
6-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N,N-dimethylpyrazin-2-amine
methyl 2-(2-{2-[(pyridin-4-ylmethyl)amino]acetamido}-1,3-thiazol-5-yl)acetate
1-[(4aR,8aS)-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-2-cyclohexylethan-1-one
[5-({[2-(1H-indol-1-yl)ethyl](methyl)amino}methyl)furan-2-yl]methanol
3-{2-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-(2,3-dichlorophenyl)-6-methylpyrimidin-2-amine
1-methyl-8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-phenyl-1,8-diazaspiro[4.5]decane
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methylbutan-1-one
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4,4,4-trifluoro-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)butan-1-one
2-hydroxy-1-[3-(3-methoxyphenoxy)azetidin-1-yl]-3-(2-methylphenoxy)propan-1-one
2,6-dimethoxy-4-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenol
(4S,4aS,8aS)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(naphthalen-1-ylmethyl)morpholine
N-cyclopropyl-4-methoxy-2-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}oxy)benzamide