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5,7-dimethyl-N-(oxan-3-yl)pyrido[2,3-d]pyrimidin-4-amine
6-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1H-pyrazol-1-yl}propanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)acetamide
1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}spiro[azepane-4,2'-chromene]
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-phenoxybutanamide
3-(2-chloro-4,6-dimethylphenyl)-1-[(3R,4R)-3-hydroxypiperidin-4-yl]urea
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(5-fluoro-2-methylphenyl)ethan-1-one
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
methyl 5-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-5-oxopentanoate
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(piperidin-3-ylmethyl)amine
N-[(4-chlorophenyl)methyl]-N-ethyl-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
10-methoxy-5-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(3S,4R)-1-[2-(1H-indol-3-yl)ethyl]-4-methylpiperidine-3,4-diol
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[1-(thiophen-2-yl)propan-2-yl]amine
ethyl 4-[(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
2-[3-(2-methoxyethyl)-5-(5-methyl-2-phenylfuran-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-[3-(pyridin-4-yl)propyl]-1H-1,2,3-benzotriazole-5-carboxamide
(1S,4R)-2-{[1-(2-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
ethyl 2-(4-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}morpholin-3-yl)acetate
(2S,4S)-N-ethyl-1-(furan-2-ylmethyl)-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
1-[1-(3-phenylpropyl)piperidin-4-yl]-N-(thiolan-3-yl)piperidine-4-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(1,3-thiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[(2,2-dimethylpropyl)(ethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2,6-dimethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
3-(2-chlorophenyl)-1-[4-(methoxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
2-{5-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1,2,4-oxadiazol-3-yl}pyrazine
3-[(3R,4S)-4-(dimethylamino)-1-{4-[(4-methylpiperazin-1-yl)methyl]benzoyl}piperidin-3-yl]propan-1-ol
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxypropan-1-one
6-cyclopentyl-2-methoxy-3-({[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-methyl-1-{1-oxaspiro[4.4]nonan-3-yl}-4-phenyl-1H-imidazole
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(3R,4R)-4-methyl-1-(5-methyl-1,3,4-thiadiazol-2-yl)-3-(propan-2-yl)pyrrolidin-3-ol
2-[2-(4-phenylpiperazin-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-cyclopentyl-4-{[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}pyrrolidin-2-one
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
methyl 3-[2-(1H-pyrazol-1-yl)acetamido]-5-[(4,5,6,7-tetrahydro-2-benzothiophen-1-ylformamido)methyl]benzoate
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(morpholin-4-yl)butan-1-one
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-3-azaspiro[5.5]undecan-9-amine
6-oxo-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-1,6-dihydropyridine-2-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-methyl-3-(thiophen-2-yl)-1H-pyrazole
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](benzyl)methylamine
N-ethyl-1-(4-methanesulfonylbenzenesulfonyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-methyl-N-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[4-(2-{2,7-diazaspiro[4.5]decan-7-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
N-[2-(4-{[2-(2H-1,3-benzodioxol-5-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide
5-chloro-3-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
2-[(3,4-difluorophenyl)methyl]-8-(2-methoxybutanoyl)-2,8-diazaspiro[4.5]decan-3-one