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1-[3-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidine-4-carboxamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
3-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}benzonitrile
methyl 6-cyclohexanecarbonyl-2-[(3,4-difluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
7-(1-aminocyclobutanecarbonyl)-N,N-dimethyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-methyl-5-[5-(1-methyl-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]pyridin-1-ium-1-olate
1-(furan-2-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
(5-{1-[(3,4-dichlorophenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
(1S,5R)-3-cyclobutanecarbonyl-6-(3-ethoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1-(6-methoxypyridin-3-yl)-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
1-cyclopentyl-5-oxo-N-{[1-(phenoxymethyl)cyclopropyl]methyl}pyrrolidine-3-carboxamide
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[7-(4-aminopyrimidin-2-yl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
1-(2-methoxyphenyl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-4-carboxamide
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
1-{2-methoxy-4-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}amino)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
1-(2-methylpropyl)-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
N-[5-(morpholin-4-yl)pentyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]cyclopentane-1-carboxamide
(3S,5S)-1-(cyclopropylmethyl)-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
5-[1-(2-phenoxyethyl)-1H-imidazol-2-yl]-2-(pyridin-2-yl)pyrimidine
N-[(3-fluoro-4-methylphenyl)methyl]-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
2-[4-(2-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-1,2,3-triazol-4-yl)acetamide
6-cyclopentyl-N-(isoquinolin-5-ylmethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-methylpyrrolidine-2-carboxamide
2-(9H-carbazol-3-yl)-1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]ethan-1-one
3-[4-(dimethylamino)phenyl]-N-methyl-N-[2-(pyridin-4-yl)ethyl]propanamide
N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]oxolane-3-carboxamide
8-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 2-(3-oxo-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-2-yl)acetate
2-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-1,2-dihydrophthalazin-1-one
6,7-dimethyl-4-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-2H-chromen-2-one
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
2-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine-3-carbonyl}pyridine
ethyl 1-{5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopentanamine
1-(4-methoxy-2-methylphenyl)-3-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}urea
(3S,4S)-1-benzoyl-4-(naphthalen-2-yl)piperidin-3-ol
2-methanesulfonyl-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-{4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-4,6-dimethylpyridine-3-carbonitrile
7-(azepane-4-carbonyl)-N,N-dimethyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[2-oxo-2-(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)ethyl]-1,2-dihydrophthalazin-1-one
N-methyl-3-(5-methyl-1H-1,2,4-triazol-3-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine
1,3-dimethyl-N-[3-(4-methylpiperazin-1-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-{2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-(pyrrolidin-1-yl)piperidine
4-{4-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione