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1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
N-ethyl-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)benzamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-(2-ethyl-1H-imidazol-1-yl)-N-methylpropanamide
6-[(3S)-3-hydroxypyrrolidin-1-yl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
[(4-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-oxazepan-6-yl)methyl]dimethylamine
5-(2-cyclopentylpyrimidin-4-yl)-2-ethoxybenzoic acid
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(cyclohex-1-en-1-yl)ethan-1-one
ethyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3,3-dimethyl-1-[(3S,4R)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]urea
2-amino-6-(2,5-dimethylthiophen-3-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(pyridin-2-yl)prop-2-enamide
2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
2-[2-(cyclopentylamino)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
(3S,4S)-1-(1H-indol-7-ylmethyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
N,N-dimethyl-1-(2-methylpropyl)-5-[(3-phenylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
9-[(3,4-dimethoxyphenyl)methyl]-3-methyl-3,9-diazaspiro[5.6]dodecane
1-(4-methoxyphenyl)-4-[2-(propylsulfanyl)acetyl]piperazin-2-one
4-(4-fluoro-2-methylphenoxy)-1-(1H-imidazol-4-ylmethyl)piperidine-4-carboxylic acid
1-(2,5-dimethylphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
methyl 4-{[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}butanoate
methyl 2-[(2-phenylethyl)sulfamoyl]-6-(pyridin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(3,4-dimethoxyphenyl)acetamide
7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
9-methoxy-N-(3-methylbutyl)-7-oxo-3-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(4-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[4-(4-methoxy-2,5-dimethylphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]methanesulfonamide
3-({4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-(2-methylbenzoyl)-4-(2-phenoxyethyl)-1,4-diazepan-5-one
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-[(4-fluorophenyl)methyl]-3-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]propanamide
2-methyl-4-oxo-N-[(2S)-oxolan-2-ylmethyl]-1,4-dihydroquinoline-8-carboxamide
2-methyl-4-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)pyrimidine
3-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-4H-chromen-4-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(quinoxaline-5-carbonyl)piperidin-3-ol
N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
5-[(4-methylpiperazin-1-yl)methyl]-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)furan-2-carboxamide
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-{3-methyl-3H-imidazo[4,5-b]pyridin-6-yl}-1,2,4-oxadiazole
2-(4-fluorophenyl)-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}morpholine
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
N-(4-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenyl)acetamide
4-(2-methoxyphenyl)-2-[5-methyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
(2S,4R)-4-amino-1-[(2,6-dimethoxyphenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
[(5-ethylpyridin-2-yl)methyl](methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-(oxolan-2-ylmethyl)-1-[1-(quinolin-2-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
N-[(3R,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-propylpyrrolidin-3-yl]-2-(methylsulfanyl)acetamide