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(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[4-(3-fluorophenyl)benzoyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
(3S,4R)-4-(2-methoxyphenyl)-1-(quinolin-8-ylmethyl)pyrrolidine-3-carboxylic acid
1-(3-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)ethan-1-one
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(1,3-thiazol-2-yl)-decahydro-1,6-naphthyridin-2-one
3-[2-amino-4-methyl-6-(3-phenylpiperazin-1-yl)pyrimidin-5-yl]propanoic acid
4-fluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-methylbenzamide
2-(2-chloro-4-{3-methyl-6-oxo-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)acetamide
({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(methyl)[1-(pyridin-2-yl)ethyl]amine
methyl 5-{[(6-methylpyridin-2-yl)methyl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(morpholin-2-yl)acetamide
1-{1-[6-(hydroxymethyl)pyridine-2-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
N-{[(2S,4S)-1-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-4-fluoropyrrolidin-2-yl]methyl}acetamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
1-(3-methylbutyl)-3,8-bis(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-hydroxy-2,2-dimethylpropyl)-6,8-dimethyl-3,4-dihydroquinazolin-4-one
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
(3R,4S)-1-(2-chloro-3-methylbenzoyl)-3,4-dimethylpiperidin-4-ol
5-(azocane-1-carbonyl)-1-(2-phenylethyl)piperidin-2-one
(4aS,8aR)-6-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-amino-2-methyl-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
1-[2-(1-{[3-(2-aminoethyl)phenyl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
2-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}azetidin-3-yl)pyridine
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3-phenyl-1,2-oxazole-5-carboxamide
5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-2-(propylsulfanyl)pyrimidine
3-[4-(dimethylamino)azepane-1-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
[(3R,4R)-1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
2-phenyl-1-(1-{spiro[2.3]hexan-1-ylmethyl}piperidin-4-yl)ethan-1-ol
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-(1H-imidazol-2-yl)piperidine
(1S,5R)-3-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 2-hydroxy-5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}benzoate
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(piperidin-1-yl)propanamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(1,3-thiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[2-(methylamino)pyridine-4-carbonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(4,4,4-trifluorobutyl)amine
N-{4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutyl}acetamide
N-cyclopentyl-5-[4-(furan-2-yl)benzoyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-[(2,3,6-trifluorophenyl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[3-(3,4-dimethoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-3-ol
5-(4-chloro-1H-pyrazole-3-carbonyl)-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2S)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}pyrrolidine-2-carboxamide
5-(2-{[(4-chlorophenyl)methyl]amino}ethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[(2-fluorophenyl)methyl]piperidine
4-ethyl-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-amino-N-(propan-2-yl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
2-{[2-(2-carboxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-1,3-oxazole-4-carboxylic acid
2-[2-(1H-imidazol-4-yl)ethyl]-8-(3-methoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
3-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
(1S,5R)-3-benzyl-6-(2,3-difluoro-4-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane