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1-(2,1,3-benzothiadiazol-5-ylmethyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-methoxy-2,2-dimethylpropan-1-one
2-{2-[1-(1,3-benzothiazole-6-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1-(2-cyclopropylphenyl)-3-[(3R)-pyrrolidin-3-yl]urea
N-[1-(1-{3-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
N-methyl-2-(2-phenylethyl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,3-benzoxazole-5-carboxamide
3-[(3R,4S)-1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
9-(5-hydroxypyrazine-2-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(morpholin-4-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 2-(piperidine-1-sulfonyl)-6-(quinolin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
2-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-3,5-dimethyl-1,4-dihydropyridin-4-one
1-(2-methoxyethyl)-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1-(1,3-thiazol-2-ylmethyl)urea
3-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-1-methyl-1H-indole
(3aS,6aS)-2-[(5-chlorofuran-2-yl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{3-ethyl-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methanol
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3R,4R)-1-(8-fluoroquinoline-2-carbonyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
4-benzyl-3-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonane
5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
N-(3-acetylphenyl)-3-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide
4-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-1,2-oxazole-5-carboxamide
3-methyl-5-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-2-yl]-1,2-oxazole
N3-methyl-N5-(2-methylpropyl)-4-oxo-N3-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[(1-benzylpiperidin-4-yl)amino]-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
N-[(2R,3R)-1'-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
3-(4-methoxyphenyl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-3-phenylpropanamide
2-(3-fluorophenyl)-N-(4-{4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}phenyl)acetamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(4-hydroxypiperidin-1-yl)acetamide
5-{2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}-1,2-dihydropyridin-2-one
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
4-[(2,5-dimethoxyphenyl)methyl]-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-methoxyethyl)-N-methyl-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]pyrrolidin-2-yl}pyridine
(3S)-1-[1-methyl-5-(thiomorpholine-4-carbonyl)-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
(2S,4S)-4-amino-N,N-diethyl-1-[2-(pyrazin-2-yl)acetyl]pyrrolidine-2-carboxamide
(3aS,6aS)-2-(2,1,3-benzothiadiazole-4-sulfonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2-{2-[1-(3,4-dimethoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine