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N3-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperidine-1,3-dicarboxamide
7-(2-chlorobenzenesulfonyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
5-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
N-{4-methyl-2-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamido]phenyl}pentanamide
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]morpholine-2-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-3-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methoxyphenyl)methyl]piperidine
1-[4-(2-methoxyphenyl)-3-oxopiperazine-1-carbonyl]cyclopropane-1-carboxamide
2-(2-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}phenoxy)ethan-1-ol
(3S,4R)-1-[2-(diethylamino)ethyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-(2-methoxyethyl)-4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine
(4aS,7aR)-1-(5-methylpyrazine-2-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(5-fluoro-2-methoxyphenyl)-3-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}urea
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(3-hydroxypiperidin-1-yl)acetamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(thian-4-yl)benzamide
methyl(2-methylpropyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
1-{2-[(cyclobutylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-4-(3-methylphenoxy)piperidine
(3aR,6aR)-2-(furan-3-carbonyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(3-chlorophenyl)methyl]-N-[2-(propan-2-yloxy)ethyl]-1,3-benzoxazole-6-carboxamide
N-[4-methoxy-3-(methylcarbamoyl)phenyl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-6-methylpyridine-3-carbonitrile
methyl 4-[6-amino-5-cyano-4-(4-hydroxy-2-methoxyphenyl)pyridin-2-yl]-5-methylfuran-2-carboxylate
(2S,4S)-4-amino-1-(2-{[5-(furan-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetyl)-N-methylpyrrolidine-2-carboxamide
4-{[4-(furan-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-3-(4-methoxyphenyl)-1H-pyrazole
methyl (2S,4S)-1-[(3-fluorophenyl)methyl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
2,3-dimethyl-7-[2-(3-phenylpyrrolidin-1-yl)acetyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazine
1-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidine-2,6-dione
4-[(4-methanesulfonylphenyl)methyl]-2-(2-methoxyethyl)morpholine
2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-(4-methylphenyl)butanamide
N-(1-hydroxyhexan-2-yl)-3-propanamidobenzamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
2-phenyl-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-ethyl-8-(pyridin-2-ylmethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
2-(3,5-difluorophenyl)-5-methyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,3-oxazole
3-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(6-methoxypyridin-3-yl)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
2-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
1-{4-[(cyclopent-3-en-1-yl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(1H-imidazol-1-yl)propan-1-one
1-{4-[(furan-2-ylmethyl)amino]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
6-cyclopropyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrimidin-4-amine
2-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-{[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
2-{1-[1-(9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
4-[4-(3-chloropyridin-2-yl)piperazin-1-yl]quinazoline
4-[2-(4-fluorophenyl)piperidine-1-carbonyl]-2-methylphenol
1-cyclopropanecarbonyl-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide