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4-{[3-(ethylcarbamoyl)pyrrolidin-1-yl]methyl}-2,6-dimethylphenyl acetate
N-(2-hydroxyethyl)-5-[(2E)-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)-1-methylpiperazin-2-one
(4aR,7aS)-1-methyl-4-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S)-1-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}pyrrolidin-3-ol
2-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-5-phenyl-2H-1,2,3,4-tetrazole
1-(1-methyl-1H-pyrazole-3-carbonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1S,5R)-6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(5-methyl-1,3-benzoxazol-2-yl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(methylsulfamoyl)ethyl]butanamide
2-[(4-methoxyphenyl)methyl]-6-(4-propylpiperazine-1-carbonyl)-1,3-benzoxazole
4-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-6-methoxypyrimidin-2-amine
methyl 3-benzamido-5-[(2,2-dimethylpropyl)amino]-1-(furan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}-3-methylpiperazin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-[(2-fluorophenyl)formamido]propanamide
1-[(6-fluoroquinolin-2-yl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-(2,5-dimethoxyphenyl)-1-(oxane-4-carbonyl)pyrrolidine
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-cyclopentyl-4-{[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]methyl}piperidine
N-(1,4-dioxan-2-ylmethyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
{4-[(2,6-difluoro-4-methoxyphenyl)methyl]morpholin-3-yl}methanol
6,7-dimethoxy-3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxylic acid
2-[4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1-(pyrrolidin-1-yl)ethan-1-one
2-(2-methoxyethyl)-8-[(4-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methylphenyl)methyl]piperidine
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1,1-dioxo-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-5-(2-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
ethyl 2-[N-methyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamido]acetate
1-({3-[1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)-1H-pyrazole
1-[2-({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-methyl-N-{4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]phenyl}furan-3-carboxamide
1-(2-cyclohexylethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-ethyl-N-[2-(thiophen-2-yl)ethyl]pyrimidine-5-carboxamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
N-(2-benzylphenyl)-3-methoxypiperidine-1-carboxamide
(3R,4R)-4-amino-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]piperidin-3-ol
3-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3,4-dihydropteridin-4-one
methyl 4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxylate
3-benzoyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
2,6-dihydroxy-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}benzamide
3,3-dimethyl-1-[(3S,4R)-1-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
1-(2-aminoethyl)-N-(2-propoxypropyl)-1H-1,2,3-triazole-4-carboxamide
1-[(1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}cyclopropyl)methyl]-1H-pyrazole
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione