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1-cyclopentyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]piperidine-3-carboxamide
8-(3-hydroxypropanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 1-{1-[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]piperidin-4-yl}piperidine-3-carboxylate
(4-{[1-(2-methyl-1,3-benzothiazole-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-[4-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-[3,5-dimethyl-4-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
(3aR,6aR)-2-[4-(dimethylamino)benzoyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]-4-(pyrimidin-2-yl)piperazine-1-carboxamide
9-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
5-{4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl}-N-methylpyrimidin-2-amine
7-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,3-diazepane-2,4-dione
1-(2-{3-[(2,6-dichlorophenyl)methyl]-1-ethyl-1H-1,2,4-triazol-5-yl}ethyl)pyrrolidin-2-one
1-cyclopentyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-[1-(4-methyl-5-phenylthiophene-2-carbonyl)azetidin-3-yl]pyridine
4-[3-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)propyl]morpholine
ethyl 2-{[5-(2-amino-3-cyano-6-cyclopropylpyridin-4-yl)pyrimidin-2-yl](methyl)amino}acetate
N-cyclohexyl-N-[(2-methylphenyl)methyl]-2-(2-oxopyrrolidin-1-yl)acetamide
4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazine-1-carboxamide
5-(2,3-dihydro-1H-indene-5-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[2-(benzylsulfanyl)ethyl]oxane-2-carboxamide
4-(2,3-dichlorophenyl)-6-methoxypyrimidin-2-amine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[(4-fluorophenyl)methyl]propanamide
4-({8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1,3-thiazole
2-ethoxy-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
6-chloro-2-methyl-4-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]quinoline
N-({1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl}methyl)furan-2-carboxamide
[3-(1H-imidazol-2-ylmethyl)-9-[(3-methylpyrazin-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
methyl 3-(furan-2-amido)-6-[(4-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
1-{4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-methoxyethan-1-one
({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
5-chloro-2-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenol
1-methyl-N-(pyridin-4-ylmethyl)-5-({[3-(trifluoromethoxy)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-6-(piperidin-3-yl)pyrimidin-4-amine
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]quinoline-2-carboxamide
5-{4-[(2-fluorophenyl)methyl]piperazin-1-yl}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(methylsulfanyl)acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-ethyl-N-[2-(pyridin-2-yl)ethyl]acetamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-[4-(piperidin-1-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]propanamide
N-ethyl-N,2-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3,3-diphenyl-1-[2-(1H-pyrazol-4-yl)ethyl]piperidine
5-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-benzylfuran-2-carboxamide
8-(3-cyclopentyl-1H-1,2,4-triazol-5-yl)quinoline
(1S,5R)-3-benzoyl-6-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
[1-(1H-indole-2-carbonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine-3-carboxamide