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2,5-dioxo-6-(pyridin-3-ylmethyl)-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[(4-methyl-5-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
N-{[(3S,4S)-1-[(6-chloropyridin-3-yl)methyl]-3-hydroxypiperidin-4-yl]methyl}-3-methylbutanamide
8-(1H-1,3-benzodiazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
3-methyl-3-phenyl-1-(1H-pyrrole-3-carbonyl)piperidine
5-[(2,3-dimethoxyphenyl)methyl]-2-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
5-acetyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]thiophene-3-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(4-fluoro-2-methylphenyl)methyl]pyrrolidin-3-yl]methanol
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(2-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
2-(1,3-dimethyl-1H-pyrazol-5-yl)-7-methyl-1H-1,3-benzodiazole
N-(1-hydroxy-2-methylpropan-2-yl)-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-ethyl-3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-1H-pyrrolo[2,3-c]pyridine-5-carboxylic acid
N-{[2-(3-methylbutyl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}benzamide
3-{[1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)pyrrolidin-3-yl]methyl}benzamide
2,2-difluoro-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
4-(1-ethyl-1H-pyrazole-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
4-methoxy-N-[4-(4-{[(4-methyl-1,3-thiazol-2-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
8-(2,2-dimethylpropyl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-6-oxo-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylacetamide
ethyl 1-(2H-1,3-benzodioxol-4-ylmethyl)-4-benzylpiperidine-4-carboxylate
4-[({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)carbamoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
4-(4-chlorophenyl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}butan-1-one
N,N-dimethyl-5-{[(3-methylphenyl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-cycloheptyl-1-(4-{[4-(3-hydroxypropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
N-methyl-N-(oxan-4-ylmethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2,5-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
1-(adamantan-2-yl)-4-[(2S,4S)-1-[(3-chlorophenyl)methyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carbonyl]piperazine
3-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)quinolin-7-ol
2-{4-[(3-ethyl-3-hydroxypiperidin-1-yl)methyl]phenoxy}acetic acid
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
3-ethyl-6-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
5-(5-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)-1H-1,3-benzodiazole
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-(2,5-dimethoxybenzoyl)-decahydro-1,6-naphthyridin-2-one
N-[(3-methoxyphenyl)methyl]-3-[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]propanamide
1-cyclopropanecarbonyl-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
4-(1H-indol-3-ylmethyl)-6-methyl-1-(2-methylphenyl)piperazin-2-one
(2-ethoxy-5-{[({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)methanol
({1-[1-(7-fluoro-4-methylquinolin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)(methyl)amine
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-methyl-4-[4-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenyl]butan-2-ol
N-[2-(2-chlorophenyl)ethyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(4-phenylpiperidin-1-yl)acetamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid