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1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
7-[(2,3-dimethoxyphenyl)methyl]-2-(3-methylbutyl)-2,7-diazaspiro[4.5]decane
2-(5-methyl-1H-pyrazol-1-yl)-1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
methyl 1-[(3S,5S)-5-(cycloheptylcarbamoyl)-1-[(2-ethoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
3-fluoro-4-methoxy-N-{2-[(2-methyl-1H-imidazol-1-yl)methyl]phenyl}benzamide
5-methanesulfonyl-1'-(pyrrolidine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(2-{4-[3-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3,4-thiadiazol-2-amine
N-[(3S,4R)-4-propyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}pyrrolidin-3-yl]acetamide
N-(2-hydroxyethyl)-1-(2-methoxyphenyl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-4-carboxamide
3-methyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-(4-cyclohexylpiperazine-1-carbonyl)-2-(pyridin-4-yl)pyrimidine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-ethyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
methyl 8-(2H-1,3-benzodioxol-4-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
6-methyl-2-{[4-(quinolin-4-yl)piperazin-1-yl]methyl}pyridin-3-ol
5-(2-amino-9H-purin-6-yl)-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)oxolane-3-carboxamide
4-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-2,2-diphenylbutanenitrile
N-[2-(4-fluorophenyl)ethyl]-3-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-ethyl-1H-indole
1-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
N'1-[(4-methoxyphenyl)(pyridin-4-yl)methyl]cyclopropane-1,1-dicarboxamide
8-[(3,5-dichloropyridin-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4S)-1-cyclopentyl-4-[2-(3,4-difluorophenyl)acetamido]-N-ethylpyrrolidine-2-carboxamide
1-tert-butyl-4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-[(3S,4R)-4-propyl-1-(quinoxalin-2-yl)pyrrolidin-3-yl]acetamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
(4aR,7aS)-1-acetyl-4-[2-(pyridin-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,6-dimethyl-N-[2-(1,3-thiazol-4-yl)ethyl]quinoline-4-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)propanamide
3-[4-(3-methoxyphenyl)phenyl]-1-methyl-1-[2-(oxan-4-yl)ethyl]urea
4-phenyl-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}azepane
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
1-(2,5-difluorophenyl)-5-[1-(ethanesulfonyl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
3-[({1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
methyl 5-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-5-oxopentanoate
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-oxo-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)piperazin-2-one
1-{2-methoxy-4-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
9-(1-benzofuran-5-ylmethyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-(1H-imidazol-4-ylmethyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-cyclopropanecarbonyl-2-(3-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3S,4R)-1-(5-fluoropyridine-3-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N,1-diethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)piperidine-4-carboxamide
1-({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)piperidine-4-carbonitrile
1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
N-(3-acetylphenyl)-3-(naphthalene-2-carbonyl)piperidine-1-carboxamide