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3-(4-fluorophenyl)-4-(1H-imidazol-2-yl)-1H-pyrazole
4-[(4-methyl-5-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-ethyl-N-[(4-methoxyphenyl)methyl]propanamide
{3-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-oxopropyl}urea
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}propanamide
3-(5-{[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,2-oxazol-3-yl)pyridine
1-[(3,5-difluoro-4-methoxyphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-11-{[(3,4,5-trifluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[(3-chlorophenyl)methyl]-N-[2-(pyridin-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-{5-[1-(2,8-dimethylquinoline-3-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
1-{3-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]phenyl}ethan-1-one
6-{1-azabicyclo[3.2.1]octan-5-yloxy}-2,3-dihydro-1H-inden-1-one
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(quinolin-6-ylmethyl)piperazin-2-yl}ethan-1-ol
3-ethyl-1-(3-methylbutyl)-8-(2-phenylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-methylpropyl)-4-[2-(4-phenylazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-(5-aminopentyl)-3-(4-fluorophenyl)-3-phenylpropanamide
6-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-9H-purine
1-ethyl-3-methyl-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-2-(2-methylphenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
2-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-2,7-diazaspiro[4.5]decane
N-[(2-chlorophenyl)methyl]-2-methanesulfonyl-N-(propan-2-yl)acetamide
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
(3S,4S)-4-cyclopropyl-1-(3-methoxy-2,2-dimethylpropanoyl)pyrrolidine-3-carboxylic acid
1-(benzenesulfonyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperazine
2-[3-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-6-(2-methoxyethyl)-3,4-dihydropyrimidin-4-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
2-(3-hydroxyphenyl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
N-(2-hydroxyethyl)-N-methyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N-(2-hydroxy-2-phenylethyl)-5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
2-methoxy-3-[3-(methoxymethyl)-1H-1,2,4-triazol-5-yl]quinoline
[1-(5-methylpyridin-2-yl)-1H-1,3-benzodiazol-2-yl]methanol
8-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1,4-dioxa-8-azaspiro[4.5]decane
N-benzyl-N-methyl-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-amine
{5-[1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
5-ethyl-1'-(1-methyl-1H-indole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 4-(5-methyl-4-{[4-(6-methylpyridin-2-yl)piperazin-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-chloro-N-[(1-ethylpiperidin-3-yl)methyl]-4-fluorobenzene-1-sulfonamide
1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(4-fluorophenyl)-1-(4-methylbenzoyl)piperidin-3-amine
8-(2,4-difluoro-3-methoxybenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3,3,3-trifluoro-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-(2-hydroxyethyl)-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
4-(dimethyl-1,2-oxazol-4-yl)-3-(1-ethoxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
({5-[1-(4-chlorobenzoyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-(2-fluorophenyl)-N-[1-(furan-2-ylmethyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
7-[2-(4-methanesulfonylphenyl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(2-fluorophenyl)ethyl)piperidin-1-yl]methyl}-3-methoxyphenol
(1r,4r)-4-[({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]cyclohexan-1-ol
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})(quinoxalin-6-ylmethyl)amine