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{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
6-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
N-(1-hydroxybutan-2-yl)-5-methoxy-N-[(2-methylphenyl)methyl]furan-2-carboxamide
3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole
2-cyclopropyl-8-(2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[(3S,4S)-3-carboxy-4-propylpyrrolidin-1-yl]sulfonyl}-1-methyl-1H-pyrrole-2-carboxylic acid
4-(1H-imidazol-1-yl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]butanamide
3-({[1-(carbamoylmethyl)piperidin-4-yl]carbamoyl}amino)-N-ethyl-2-methylbenzamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]ethan-1-one
3-acetyl-N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
4-fluoro-3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
(3S,4R)-1-[2-(azocan-1-yl)acetyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})(1,3-thiazol-4-ylmethyl)amine
N,3-dimethyl-N-[(1-methylpyrrolidin-2-yl)methyl]-5-propyl-1-benzofuran-2-carboxamide
1-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-4-methylpiperidine-4-carbonitrile
2-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-N-(1,3-thiazol-2-yl)acetamide
4-[({[3-hydroxy-2-oxo-1-(3-phenylpropyl)piperidin-3-yl]methyl}amino)methyl]benzonitrile
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-cycloheptanecarbonylpiperidin-3-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-(3,4-dimethylpiperazin-1-yl)pyrimidine
5-(pyrrolidin-1-yl)-2-(1,3-thiazol-4-ylmethyl)-2,3-dihydropyridazin-3-one
2-methoxy-1-(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]cyclopentanecarboxamide
1-{4-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]piperidin-1-yl}ethan-1-one
4-acetamido-N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N4-[(1R)-1-(4-methoxyphenyl)ethyl]-5-methylpyrimidine-2,4-diamine
3-(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)benzonitrile
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
5-cyclohexyl-3-(2,4-dimethoxyphenyl)-1H-1,2,4-triazole
4-sulfamoyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]butanamide
6-methoxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-amine
propan-2-yl 4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-(2,3-dihydro-1H-isoindol-2-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-[4-(difluoromethoxy)phenyl]-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
3,4,4-trimethyl-1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-ol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)amine
N-[(3R,4S)-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
2-oxo-3-[2-(pyridin-2-yl)ethyl]-1-[2-(1H-pyrrol-1-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
(5-methyl-3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-oxazol-4-yl)methanol
1-methoxy-3-{2-[2-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}propan-2-ol
3-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
4-(1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidin-4-yl)pyridine
8-[2-(diethylamino)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one