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2-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
3-{[2-(3-fluorophenyl)ethyl]sulfamoyl}-N-methyl-N-propylbenzamide
2-methoxy-N-[1-methyl-2-(pyridin-3-yl)-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-7-yl]acetamide
methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl][1-(pyridin-3-yl)ethyl]amine
3-(3-fluorophenyl)-4-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
2-(ethylamino)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrimidine-5-carboxamide
2-[4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)morpholin-3-yl]-N-(2-fluorophenyl)acetamide
(4aS,7aR)-1-[3-(4-fluorophenoxy)propyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopentyl-2,4-dimethyl-N-(prop-2-en-1-yl)pyrimidine-5-carboxamide
2-[4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(quinoxalin-2-yl)-1,4-diazepan-5-one
5-methyl-4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]pyrimidin-2-amine
N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
3-[3-(2-amino-3-cyano-5,6,7,8-tetrahydroquinolin-4-yl)-1H-indol-1-yl]propanamide
6,7-dimethoxy-2-[(1-methyl-1H-imidazol-5-yl)methyl]-1-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
N-(2-{4-[(2-methylphenyl)methyl]morpholin-2-yl}ethyl)cyclopropanesulfonamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]morpholine-4-sulfonamide
(4aS,8aR)-1-(pyridin-4-ylmethyl)-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-ethyl-4-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
2-{4-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-yl]methanol
3-methyl-N-[(5-methylpyrazin-2-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
2-(2-fluorophenoxymethyl)-N-(isoquinolin-5-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-methyl-4-[(3-phenylpiperidin-1-yl)methyl]benzene-1-sulfonamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(oxan-4-yl)acetamide
5-(2-chlorophenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)furan-2-carboxamide
N-[(3-methyl-7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-phenoxypropanamide
1-{4-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
1-{5-[5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}-2-(methylsulfanyl)ethan-1-one
N-benzyl-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-{1-[(1,3-dimethyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidine-2-carboxamide
(3S,9aR)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl (1R,3S,3aR,6aS)-3-(2-chloro-4-fluorophenyl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-(1H-imidazol-2-yl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
2-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]morpholin-3-yl}acetic acid
3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-N-(pyridin-3-yl)benzamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1H-1,2,4-triazole
2-(ethylamino)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}pyrimidine-5-carboxamide
1-[(1R)-2,3-dihydro-1H-inden-1-yl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-fluoro-1,3-dimethyl-1H-indole-2-carboxamide
6-methyl-2-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
3-(1-methyl-1H-pyrazol-5-yl)-N-[(3-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)propanamide
2-(3-methylbutyl)-8-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(2-phenylethyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(N-methylmethanesulfonamido)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide