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6-(3-ethoxyphenyl)pyridin-2-amine
(3R,9aR)-8-(3-chlorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-4-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}phenol
2-methyl-4-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-propylpyrimidine
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(5-methylpyridin-2-yl)pyridine-3-carbonitrile
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-(1H-indazol-7-yl)urea
4-[(3-methoxyphenyl)methyl]-1-[(1-methyl-1H-indol-3-yl)methyl]-1,4-diazepan-5-one
N-{2-[1-({[(2-fluorophenyl)methyl]carbamoyl}methyl)piperidin-2-yl]ethyl}acetamide
2-(3-acetyl-1H-indol-1-yl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}butan-1-one
N-(3-{[(2-methanesulfonamidoethyl)carbamoyl]amino}-2-methylphenyl)cyclopentanecarboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
5-{methyl[1-(thiophen-2-yl)ethyl]amino}-1-{[3-(trifluoromethyl)phenyl]methyl}azepan-2-one
(4aS,8aR)-6-(2-amino-9H-purin-6-yl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{[2-(2,3-difluorophenyl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1,3,7-trimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-indole-2-carboxamide
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-sulfonyl]-N-[(2S)-1-hydroxypropan-2-yl]benzamide
(2R,3R,6R)-5-(5-methyl-1,3-oxazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-[(2,3-dimethoxyphenyl)methyl]-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
5-(phenoxymethyl)-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
2-{[2-({[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}carbamoyl)phenyl]amino}acetic acid
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{2-oxo-1'-[3-(pyridin-4-yl)propanoyl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
1-ethyl-N,N-dimethyl-4-({[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)piperidin-4-amine
3-{[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]sulfonyl}benzoic acid
3-(3-chloro-1,2-oxazol-5-yl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-(4H-1,2,4-triazol-4-yl)-2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
(1R,9aR)-1-[(2,3-dihydro-1,4-benzodioxin-6-yloxy)methyl]-octahydro-1H-quinolizine
2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluoro-2-methoxyphenyl)acetic acid
1-(1-methyl-1H-pyrazole-5-carbonyl)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-[2-(1H-pyrazol-1-yl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
(1R,3S)-3-{[(3,4-difluorophenyl)methyl]carbamoyl}cyclopentane-1-carboxylic acid
(3aR,6aR)-2-cyclopropanecarbonyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]urea
3-[2-(2-hydroxyethoxy)ethyl]-1-[3-methyl-1-(4-methylquinolin-2-yl)-1H-pyrazol-5-yl]urea
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-(4-fluorobenzenesulfonyl)pyrrolidine
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{[methyl(propan-2-yl)amino]methyl}piperidin-2-one
3-{1-[(2,2-dimethyloxan-4-yl)methyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-[2-(2,3-dichlorophenyl)ethyl]-2-[methyl(piperidin-4-yl)amino]acetamide
1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
4-{[1-(2-hydroxyethyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
7-[(2,3-difluorophenyl)methyl]-2-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
N-(cyclobutylmethyl)-3-{imidazo[1,2-a]pyridin-2-yl}-N-(oxolan-2-ylmethyl)propanamide
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methylurea
N-{[3-(cyclopentyloxy)phenyl]methyl}-1,3-dimethyl-N-[(3S)-2-oxoazepan-3-yl]-1H-pyrazole-5-carboxamide
N5-cyclohexyl-1-cyclopropyl-N3-methyl-4-oxo-N3-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-hydroxyethan-1-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]acetamide
2-{[(3-methoxypyrazin-2-yl)(methyl)amino]methyl}-3,4-dihydroquinazolin-4-one