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(3aS,6aS)-2-cyclopropanecarbonyl-5-[(2-methylpropoxy)carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-6-[1-(methylsulfanyl)propan-2-yl]-3-(quinolin-6-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-3-(piperidin-3-yl)benzamide
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-hydroxyazepan-4-yl]methyl}furan-2-carboxamide
3,5-dimethyl-2-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-indole
1-methyl-6-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
3-(1H-pyrazol-1-ylmethyl)-N-[1-(thiophen-2-yl)ethyl]benzamide
N-[1-(2-methylphenoxy)propan-2-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
2-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
2-{5-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-ethyl-8-{2-[4-(trifluoromethyl)phenyl]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
(1S,6R)-9-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-ethylpyrrolidin-2-one
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
8-[3-(2-methoxyphenyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 1-[(4-acetamidophenyl)methyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-amino-6-(2,2-dimethylcyclopropyl)-4-(4-hydroxy-3,5-dimethoxyphenyl)-5-methylpyridine-3-carbonitrile
N-({1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]piperidin-4-yl}methyl)acetamide
4-[1-(3-methylbutyl)-5-{[4-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
2-(dimethylamino)-7-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(2-{[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-{4-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperazin-1-yl}benzoic acid
2-(4-hydroxypiperidin-1-yl)-N-[2-(3-phenylpropoxy)phenyl]acetamide
ethyl 2-[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]acetate
(3aS,6aS)-3a-(hydroxymethyl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)-octahydrocyclopenta[c]pyrrole-2-carboxamide
1-{4-[(butylamino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-[methyl(phenyl)amino]acetamide
1-(2-methoxyethyl)-3-[(2-methylphenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-[7-(hydroxymethyl)-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-methoxyethan-1-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-(4-methylphenyl)-3-phenylpropanamide
(1S,3R)-N1-[(2-ethoxyphenyl)methyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methylpropanamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(5-acetylthiophen-3-yl)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]acetamide
(2S,4R)-4-amino-N-ethyl-1-(5-methyl-1H-1,3-benzodiazole-2-carbonyl)pyrrolidine-2-carboxamide
2-cyclopropyl-N-[3-(1H-indazol-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-2-(2,3-dihydro-1H-inden-1-yl)ethan-1-one
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-(pyridin-2-yl)acetamide
(3aR,6aR)-2-acetyl-5-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-benzyl-8-[(4-hydroxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-{1-cyclohexyl-5-[2-(pyrazin-2-yl)ethyl]-1H-1,2,4-triazol-3-yl}benzamide
2-{4-[(3-chloro-1-benzothiophen-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
(3S,4R)-1-(1-benzyl-5-methyl-1H-1,2,3-triazole-4-carbonyl)-3-methoxypiperidin-4-amine
[1-(dimethylamino)propan-2-yl]({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl})amine
2,2,2-trifluoro-N-{2-[(3-methyl-1-benzothiophen-2-yl)formamido]ethyl}acetamide
3,5-dimethyl-2-{[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,4-dihydropyridin-4-one
3-{5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid