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1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
4-(cyclobutylmethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(2H-1,2,3-benzotriazol-2-yl)-1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}ethan-1-one
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-(4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}phenoxy)pyrimidine
2-{4-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]-1-(cyclopropylmethyl)piperazin-2-yl}ethan-1-ol
5-(5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,2,4-oxadiazol-3-yl)-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-benzyl-N-methyl-2-(morpholin-4-ylmethyl)piperidine-1-sulfonamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine
N-cyclopropyl-6-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-{4-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-[(2-chlorophenyl)methyl]-4-(pyrimidin-2-yl)morpholine
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}azepan-4-amine
2-[(3,4-dimethoxyphenyl)methyl]-6-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,3-benzoxazole
1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (1R,3S,3aR,6aS)-5-ethyl-4,6-dioxo-3-(2,4,5-trifluorophenyl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(3R,4R)-1-{[3-(furan-2-yl)phenyl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(3,3,3-trifluoropropanoyl)-2,8-diazaspiro[4.5]decan-3-one
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-[(2-propyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-cyclopropyl-1-{2-[1-(2-phenoxyacetyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-{1-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
3-methyl-7-{[4-(pyridin-3-yl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-{[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
8-(3-methyl-5-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-1,2,4-triazol-1-yl)quinoline
4-[(2,3-dihydro-1,4-benzodioxin-5-yloxy)methyl]-2-(furan-2-yl)-5-methyl-1,3-oxazole
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[3-(pyridin-3-yl)propyl]amine
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(2-oxopyrrolidin-1-yl)propanamide
3-benzoyl-1-(2,3-dihydro-1H-indene-5-carbonyl)piperidine
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](furan-2-ylmethyl)amino}butan-1-ol
1-{3-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
benzyl 4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxylate
2-(1-tert-butyl-1H-pyrazol-4-yl)-N,7,8-trimethyl-N-(propan-2-yl)quinoline-4-carboxamide
3-{4-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperazin-1-yl}propan-1-ol
ethyl 4-benzyl-1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidine-4-carboxylate
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-3-[2-(1H-imidazol-1-yl)propyl]urea
methyl 6-cyclopentanecarbonyl-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(7R,9aR)-N-cyclohexyl-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
[1-(2,5-dimethylfuran-3-carbonyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
1-[(2-chloro-6-fluorophenyl)methyl]-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1H-1,2,4-triazole
6-(benzyloxy)-1-cyclohexyl-4-(pyridine-3-carbonyl)-1,4-diazepan-2-one
3-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-4-ol
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
1-[(6-ethyl-2-oxo-2H-chromen-4-yl)methyl]piperidine-3-carboxamide
N-[2-(5-methylfuran-2-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide