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N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-methyl-5-{[(5-methylfuran-2-yl)methyl]amino}-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(4aS,8aR)-6-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
6-methyl-4-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-3-carboxamide
3-{3-[1-(dimethylamino)ethyl]phenyl}-5-hydroxybenzoic acid
2-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}pyridine-4-carboxamide
4-methyl-6-(1H-pyrazol-4-yl)-2-(pyrrolidin-1-yl)pyrimidine
(4S)-3-{2-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
5-[4-(4-fluorophenyl)piperazin-1-yl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(1-methylpiperidin-4-yl)piperazine
2-(2-methoxy-5-methylphenyl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
(4aS,8aR)-2-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-decahydroisoquinoline
2-(4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-[2-(dimethylamino)ethyl]-N-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
4-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-phenylpiperazin-2-one
6-(benzyloxy)-4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(1-methyl-1H-pyrazol-5-yl)propanamide
{1-[1-(4-chloro-1-methyl-1H-indole-2-carbonyl)piperidin-3-yl]piperidin-4-yl}methanol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
{2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-8-methylquinolin-3-yl}methanol
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl][(3-methylthiophen-2-yl)methyl]amine
2-(furan-2-ylmethyl)-3-[(5-methylpyrimidin-2-yl)amino]propan-1-ol
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-3-(3-methylphenoxymethyl)piperidine
5-ethyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-ethyl-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
N'-cycloheptyl-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)butanediamide
1-[(2-{1-butyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]-1H-pyrazole
2-{4-[1-(naphthalen-1-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
5-methyl-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)propanamide
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
5-methyl-4-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,3-oxazole
2-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-2-azaspiro[4.5]decan-3-one
1-methyl-8-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)quinoline-4-carboxamide
N6-cyclopentyl-N5-methyl-N5-(pyridin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(dimethylamino)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(4-methylphenyl)acetamide
N-(4-cyanophenyl)-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}benzamide
N-[2-(diethylamino)ethyl]-N,1-dimethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}furan-2-yl)methyl]morpholine
2-({5-[2-methoxy-5-(propan-2-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}methyl)-5-methyl-1,3,4-oxadiazole
1-methyl-3-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-(3-phenylpropyl)-4-(thiophene-3-carbonyl)morpholine
1-ethyl-4-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}piperazine-2,3-dione
3-{1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-pyrazol-4-yl}benzoic acid
9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one