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(3R,4R)-1-(cyclopentylmethyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
(2S,4R)-4-amino-N-methyl-1-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]pyrrolidine-2-carboxamide
2-[(furan-2-ylmethyl)({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]butan-1-ol
2-methoxy-4-[3-(2-methoxyphenoxy)azetidin-1-yl]pyridine-3-carbonitrile
methyl 1-[9-methoxy-3-(2-methylpropyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
5-butyl-N4-[(4,6-dimethylpyrimidin-2-yl)methyl]-6-methylpyrimidine-2,4-diamine
N-(2H-1,3-benzodioxol-5-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-amine
N-benzyl-1-[(2-chlorophenyl)methyl]-N-(cyclobutylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-ethyl-3-methyl-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-N-(thiophen-2-yl)piperidine-1-carboxamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]urea
3-[(dimethylamino)methyl]-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-ol
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N,N-dimethylpyridine-3-carboxamide
ethyl 2-(4-{9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carbonyl}morpholin-3-yl)acetate
5-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-1-[(4-methylphenyl)methyl]azepan-2-one
5-methyl-N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
4-cyclopentyl-N-[1-(3-methylpyridin-2-yl)propyl]pyrimidin-2-amine
(4aR,8aR)-7-(3-cyano-2-methoxypyridin-4-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
1-tert-butyl-N-[3-(4-fluorophenyl)propyl]-5-oxopyrrolidine-3-carboxamide
N-[(2-methoxyphenyl)methyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-propylbenzamide
3-{1-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
2-(5-{[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}furan-2-yl)benzonitrile
1-(4-{2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethoxy}phenyl)propan-1-one
1-({5-[(1-ethyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
1-(3-chlorophenyl)-4-[1-(3-methylbutyl)piperidin-3-yl]piperazine
3-(1H-indol-5-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
3-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
(3S,4S)-1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
1-[3-(1H-pyrazol-1-yl)propyl]-1,2-dihydroquinoxalin-2-one
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(4aS,7aR)-1-(furan-3-ylmethyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(5S,9aS,9bS)-2-phenyl-5-(quinolin-8-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[2-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)phenoxy]acetic acid
4-methoxy-N-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-[(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]-2-methylpropanamide
5-[({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)sulfanyl]-1,3,4-thiadiazol-2-amine
2-cyclohexyl-N-[2-(dimethylsulfamoyl)ethyl]-1,3-benzoxazole-6-carboxamide
N-{4-[1-(2-hydroxyethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]phenyl}ethane-1-sulfonamide
2-methyl-N-[2-(5-methylthiophen-2-yl)ethyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
5-[methyl(thiophen-3-ylmethyl)carbamoyl]-1H-imidazole-4-carboxylic acid
1-[(5-ethylfuran-2-yl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
(2R,3R,6R)-5-[(2-ethylpyrimidin-4-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(4-fluorophenyl)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-(2-cyclohexylethyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-(1H-pyrazol-1-ylmethyl)-4-[4-(trifluoromethyl)pyrimidin-2-yl]-1,4-oxazepane
1-methyl-5-[2-(2-phenylethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
8-[(4-fluorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methyl-4-[4-(1-methylpiperidin-4-yl)piperazine-1-carbonyl]quinoline
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N,N-bis(prop-2-en-1-yl)acetamide