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3-(1,3-benzoxazol-2-yl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
2-(azocan-1-yl)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one
5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]-3-propyl-1,2,4-oxadiazole
3-(1H-imidazol-2-yl)-6-methyl-4H-chromen-4-one
7-(3-chlorophenyl)-4-[(3-ethyl-1H-pyrazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[4-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(piperidine-1-carbonyl)pyridine
4-methoxy-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}benzamide
1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(thiophene-2-carbonyl)piperazine
1-[2-methoxy-5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
5-fluoro-4-methoxy-2-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]pyrimidine
N-methyl-2-{4-[(E)-2-phenylethenyl]phenyl}acetamide
4-[5-(methoxymethyl)furan-2-carbonyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-cyclopropyl-N-[(3-methoxyphenyl)methyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]piperidine-4-carbonitrile
3-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]-4-(cyclohexylmethyl)piperazin-2-one
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-2,5-dimethoxybenzamide
2-[benzyl({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
5-[4-(3-methylphenyl)piperazine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
2-ethyl-4-({4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
2,6-dimethoxy-N-[1-(pyridin-2-yl)propan-2-yl]pyridine-3-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(4-methylquinolin-2-yl)pyrrolidin-3-yl]acetamide
1-{[3-(benzyloxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
4,4-difluoro-N-(2-fluoro-5-methylphenyl)piperidine-1-carboxamide
(1R,5R)-3-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-8-propyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-[(5-fluoro-2-methoxyphenyl)methyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
5-{[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]methyl}-3-methyl-1,2-oxazole
(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-7-{[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(propan-2-yl)thiophene-3-carboxamide
N,N-diethyl-1-[(1s,4s)-4-(2,2-dimethylpropanamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-methoxy-N-[4-methyl-2-(pyrimidin-5-yl)phenyl]benzamide
N,5-dimethyl-2-(2-methylpropanamido)-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-3-(4-methylpiperazine-1-carbonyl)-1,4-dihydropyridin-4-one
methyl (2S,4S)-1-[(2-chlorophenyl)methyl]-4-(pyridine-2-amido)pyrrolidine-2-carboxylate
1-benzyl-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
2-(6,8-dichloro-4-oxo-3,4-dihydroquinazolin-3-yl)-N-methylacetamide
methyl 4-(2-chloro-3,4-dimethoxyphenyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
1-ethyl-4-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}piperazine
3-{5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
(2R)-2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-methylbutanamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-amine
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-({4-[5-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)quinolin-7-ol
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
2-(2,6-difluorobenzenesulfonyl)-8-methyl-2,8-diazaspiro[4.5]decane
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one