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4-(2,6-dimethylpyridin-3-yl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-2-amine
1-(4-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)imidazolidin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[3-(propan-2-yloxy)phenyl]-4-(pyrrolidine-1-carbonyl)pyridine
8-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(2-oxopyrrolidin-1-yl)butanamide
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-N-(2-methylpropyl)acetamide
[(1-cyclohexylpiperidin-3-yl)methyl](cyclopropylmethyl)(pyridin-3-ylmethyl)amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl})amine
6,7-dimethyl-4-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)-2H-chromen-2-one
N-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-{[2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N-(4-oxo-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butyl)acetamide
(4aR,7aS)-1-acetyl-4-(1-ethyl-1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 8-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[3-(2,5-difluorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
N-ethyl-2-(4-{2-[(1-ethyl-1H-indol-3-yl)sulfanyl]acetyl}morpholin-3-yl)acetamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-(2,3,6-trifluorophenyl)ethan-1-one
(1H-indol-2-ylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
1-(azepan-1-yl)-4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]butane-1,4-dione
N-[1-(pyridin-2-yl)propyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
3-{[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}-1-(pyrrolidin-1-yl)propan-1-one
1-{2-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,2-dihydroquinoxalin-2-one
N-(3,4-dimethylphenyl)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
2-amino-4-[6-(dimethylamino)pyridin-3-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1-(3-carbamoylpyridin-2-yl)-4-phenoxypiperidine-4-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(furan-2-yl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidin-2-yl)pyridine
1-[(2-fluoro-4-methoxyphenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-ethyl-5-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
(1R,5R)-6-(1-benzothiophene-2-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
6-methyl-4-oxo-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-4H-pyran-2-carboxamide
2-({4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)pyrimidine
3-({1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidin-4-yl}oxy)pyridine
N,N-dimethyl-2-{[(3-phenyl-1,2,4-oxadiazol-5-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[(3-fluorophenyl)methyl]-4-[2-(morpholin-4-yl)butanoyl]piperazin-2-one
2-butyl-8-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-2-cyclobutyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-fluoro-2-methoxy-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(2-methylphenyl)pyrrolidin-3-ol
(2S)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-(2-{2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}ethyl)piperidine
1-(4-methyl-2-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}pyrimidin-5-yl)ethan-1-one
N-(2,2-dimethyloxan-4-yl)-4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-ethylpyrimidin-2-yl)piperidin-3-ol
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]propanamide
4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-2-(propan-2-yl)pyrimidine
4-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
5-[5-(3,5-dimethyl-1-benzofuran-2-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole