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1-(4-chloro-2-methoxy-5-methylphenyl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
N-[3-({[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
1-ethyl-N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1H-pyrazole-4-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-2-fluoro-5-sulfamoylbenzamide
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyacetyl)pyrrolidin-3-yl]methanesulfonamide
(1S,5R)-6-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-methylpropanamide
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-N,N-dimethylaniline
[(4-cyclopropyl-5-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
3-{6-amino-5-cyano-4-[2-(propylamino)pyrimidin-5-yl]pyridin-2-yl}-1H-pyrazole-5-carboxylic acid
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyridin-4-ylmethyl)piperazine
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[2-(3-cyano-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)ethyl]-2-methylpropanamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-7-fluoro-3-methyl-1-benzofuran-2-carboxamide
6-(2-chlorophenyl)-N-methyl-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(aminomethyl)-4-[(1R)-1-(4-methoxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(methoxymethyl)-5-({8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)pyrimidine
methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)(1,3-thiazol-2-ylmethyl)amine
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(pyridin-3-yl)propanamide
1-methyl-2-oxo-8-(4-phenoxybutanoyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(3-methoxypropyl)-2-methyl-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}propanamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2,4-dichloro-5-fluorophenyl)methyl]-5-methylpyrrolidin-2-one
1-(1H-indol-3-ylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}benzamide
1-(4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}piperidin-1-yl)-2-methoxyethan-1-one
6-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]ethan-1-one
N-[2-(3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenoxy)propyl]-2-(thiophen-3-yl)acetamide
1-{3-[(4-fluoropiperidin-1-yl)methyl]-6-methylquinolin-2-yl}piperidin-3-ol
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-(1H-pyrazol-5-ylmethyl)benzamide
N-ethyl-N-propyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-(cyclohex-3-ene-1-carbonyl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
3-(2H-1,3-benzodioxol-5-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
4-(2-cycloheptylethyl)-2-ethyl-1-methylpiperazine
(2S)-4,4-difluoro-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidine-2-carboxamide
2-(1-methyl-1H-imidazol-5-yl)-1-[2-(oxolan-2-ylmethoxy)phenyl]-1H-imidazole
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(4,4,4-trifluorobutyl)piperidine-2-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-propylpyrimidine-5-carboxamide
1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazole
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-5-(methoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]furan-2-carboxamide
(3S,4S)-1-{2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carbonyl}piperidine-3,4-diol
[(3R,4R)-4-[(dimethylamino)methyl]-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]pyrrolidin-3-yl]methanol
2-{2-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-fluorophenyl)methyl]-1-methyl-1H-pyrazole-5-carboxamide
(2S,4R)-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)-4-[(pyridin-3-ylmethyl)amino]pyrrolidine-2-carboxamide
7-(2,7,8-trimethylquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one