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N-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)phenyl]acetamide
3-cyclopropyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
N-ethyl-3-{[3-(2-fluorophenyl)propyl]sulfamoyl}-N-methylbenzamide
1-benzyl-3-methyl-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(1-tert-butyl-1H-pyrrole-3-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-methoxyphenyl)methyl]-3-(1-phenylmethanesulfonylpiperidin-3-yl)propanamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[4-(pyridin-2-yl)butyl]amine
5-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methoxyphenol
(3R,4S)-4-(5-methylfuran-2-yl)-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-amine
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2-(thiophen-2-yl)pyrimidine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methoxypyrimidin-2-amine
1-({3-[2-(methylsulfanyl)ethyl]-1-propyl-1H-1,2,4-triazol-5-yl}methyl)-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-(cyclopropylmethyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-methyl-2-[1-(propan-2-yl)piperidin-4-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
1-cyclopropyl-N-[3-(4-fluorophenyl)propyl]-5-oxopyrrolidine-3-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
(2R,6S)-4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2,6-dimethylmorpholine
N-[3-(4-methylbenzamido)phenyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
3-methoxy-1-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
1-[4-(thiomorpholine-4-sulfonyl)benzoyl]pyrrolidin-3-ol
N-cyclohexyl-5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
5-(2,6-dimethylquinoline-4-carbonyl)-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-[3-(pyridin-4-yl)propyl]-6-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)propanamide
2-phenyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}pyrimidine-5-carboxamide
3-butyl-1-methyl-4-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)piperazin-2-one
N-[(2-fluorophenyl)methyl]-2-(N-phenylmethanesulfonamido)propanamide
{5-methyl-7-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
[(1-cyclopentylpiperidin-4-yl)methyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-(4-ethyl-1H-pyrazol-5-yl)-1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidine
3-{4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
4,5-dimethyl-6-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}pyrimidine
3-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2-dihydroquinoxalin-2-one
1-(9H-purin-6-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}piperidin-4-amine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-cycloheptyl-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl})amine
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(isoquinolin-5-ylmethyl)-N-methylpyrazin-2-amine
1-(morpholin-4-yl)-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-N-(2-methoxyethyl)-3-methylbenzamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[(2-phenoxyethyl)amino]methyl}piperidin-2-one
2-fluoro-N-{3-[4-(3-methylpyridin-4-yl)piperazin-1-yl]-3-oxopropyl}benzamide
8-(2-ethoxyethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-4-(piperidin-4-yl)-6-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrimidine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(piperidin-4-yl)piperidine-4-carboxamide
4-{1-[1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine